Target Details
| UniProt AC | P09769 |
|---|---|
| Gene Symbol | FGR |
| Protein Name | Tyrosine-protein kinase Fgr |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 96
- Clinical molecules 21
- Avg pChEMBL 7.09
KEGG Pathways (1)
Active Molecules (96)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
6.9 | Kd | 231 | Yes | |
OSAWFUCUZJNEID
|
6.9 | IC50 | 20 | — | |
ZZSBPGIGIUFJRA
|
6.8 | Kd | 46 | — | |
RNOAOAWBMHREKO
|
6.8 | IC50 | 15 | — | |
MFAQYJIYDMLAIM
|
6.8 | Kd | 130 | Yes | |
ZTUJNJAKTLHBEX
|
6.7 | IC50 | 5 | — | |
OYKPWSZSBLRRPL
|
6.7 | IC50 | 11 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
PIQCTGMSNWUMAF
|
6.7 | Kd | 137 | Yes | |
VTJHGMZHVOXJPG
|
6.7 | IC50 | 15 | — | |
GUBJNPWVIUFSTR
|
6.7 | Kd | 103 | — | |
HHFBDROWDBDFBR
|
6.7 | Kd | 40 | Yes | |
UHIZYQVRKSWIFO
|
6.6 | Kd | 3 | — | |
WMMNTQFZCHUZSM
|
6.6 | IC50 | 14 | — | |
UHTHHESEBZOYNR
|
6.6 | Kd | 66 | Yes | |
WDTHDWKPTWWHLS
|
6.6 | IC50 | 13 | — | |
WINHZLLDWRZWRT
|
6.6 | Kd | 201 | Yes | |
XZXHXSATPCNXJR
|
6.5 | Kd | 165 | Yes | |
HHZIURLSWUIHRB
|
6.5 | Kd | 57 | Yes | |
GLBZSOQDAOLMGC
|
6.5 | IC50 | 23 | Yes | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
ZATGFXTWDKIEKC
|
6.4 | IC50 | 8 | Yes | |
UKYJKXMPIDEQFF
|
6.4 | IC50 | 16 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
APPXQUDJLJXULP
|
6.3 | IC50 | 47 | — | |
AILRADAXUVEEIR
|
6.3 | IC50 | 75 | — | |
AKSZNKRUJCTEIJ
|
6.3 | IC50 | 4 | — | |
CDBACQLZGUZJLV
|
6.3 | IC50 | 2 | — | |
NKTVKMCHRMDFHV
|
6.3 | IC50 | 5 | — | |
QZCWPDPWSBOTEU
|
6.3 | IC50 | 7 | — | |
RSWVUHGRSKMXFQ
|
6.3 | IC50 | 3 | — | |
RITAVMQDGBJQJZ
|
6.2 | Kd | 43 | — | |
WJEOLQLKVOPQFV
|
6.2 | Kd | 24 | — | |
RMTJSBZCZKCYHB
|
6.2 | IC50 | 13 | — | |
KTEIFNKAUNYNJU
|
6.2 | Kd | 114 | — | |
YOVVNQKCSKSHKT
|
6.2 | IC50 | 15 | — | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 91 | Yes | |
UORAPQCBWYIISR
|
6.1 | IC50 | 15 | — | |
UORAPQCBWYIISR
|
6.1 | IC50 | 13 | — | |
GCIKSSRWRFVXBI
|
6.1 | Kd | 109 | Yes | |
OUKYUETWWIPKQR
|
6.0 | Kd | 31 | Yes | |
WVUNYSQLFKLYNI
|
6.0 | Kd | 46 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |