Target Details
| UniProt AC | P09769 |
|---|---|
| Gene Symbol | FGR |
| Protein Name | Tyrosine-protein kinase Fgr |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 96
- Clinical molecules 21
- Avg pChEMBL 7.09
KEGG Pathways (1)
Active Molecules (96)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SFCBIFOAGRZJNX
|
9.5 | Kd | 22 | — | |
SSDFTYWIYVWCIE
|
9.4 | IC50 | 17 | — | |
ZBNZXTGUTAYRHI
|
9.3 | Kd | 102 | Yes | |
WFRLFWGASBLYTC
|
9.1 | IC50 | 15 | Yes | |
FZBVNCFBCNXULH
|
8.7 | IC50 | 18 | — | |
LCYSSHSIKSARGO
|
8.6 | IC50 | 19 | — | |
XYFPWWZEPKGCCK
|
8.6 | IC50 | 34 | — | |
VAARYSWULJUGST
|
8.6 | Kd | 119 | Yes | |
UBPYILGKFZZVDX
|
8.6 | IC50 | 130 | Yes | |
ZCWXCBKGPJOAFQ
|
8.4 | IC50 | 13 | — | |
XHKFYFCKCXKVPO
|
8.3 | IC50 | 5 | — | |
CIGMIXWAESLRNR
|
8.2 | Kd | 5 | — | |
MIMOHMCANSGXIG
|
8.0 | IC50 | 15 | — | |
IRBVGTPPFBYDKX
|
7.8 | IC50 | 9 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 213 | — | |
AYCPARAPKDAOEN
|
7.7 | IC50 | 73 | — | |
LSJWYMSFUWBGPN
|
7.7 | IC50 | 17 | — | |
CDISOBGWDHAHGF
|
7.6 | IC50 | 16 | — | |
KCPKCAYWGNEVBR
|
7.6 | IC50 | 7 | — | |
LXURGGKEOPHREO
|
7.5 | IC50 | 13 | — | |
OPHSZSZDICRBPP
|
7.5 | IC50 | 16 | — | |
NHHQJBCNYHBUSI
|
7.5 | Kd | 220 | — | |
QHXBWJSQXSYAGG
|
7.5 | IC50 | 16 | — | |
FUZSHLVNKZZEKR
|
7.5 | IC50 | 16 | — | |
JUSWPUDQOKINJO
|
7.4 | IC50 | 16 | — | |
PHXJVRSECIGDHY
|
7.4 | Kd | 59 | — | |
WVXNSAVVKYZVOE
|
7.4 | IC50 | 92 | — | |
GZYUJXFTHLKPAK
|
7.4 | IC50 | 16 | — | |
CXQHYVUVSFXTMY
|
7.4 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.4 | Kd | 149 | — | |
CEUSZLVORFRBCV
|
7.4 | IC50 | 13 | — | |
PTHVKCSYXICMAR
|
7.4 | IC50 | 14 | — | |
GMVQPWCWWLPOQT
|
7.4 | IC50 | 9 | Yes | |
UIARLYUEJFELEN
|
7.3 | Kd | 289 | Yes | |
UORAPQCBWYIISR
|
7.3 | IC50 | 12 | — | |
KUCNBQPAJZRQMJ
|
7.3 | IC50 | 11 | — | |
KZRDVFBPXXGSPD
|
7.3 | IC50 | 9 | — | |
MJQGHLODJHABRA
|
7.3 | IC50 | 10 | — | |
QUFURWJAQILIFO
|
7.3 | IC50 | 9 | — | |
XYFZVVYVIFJBIS
|
7.3 | IC50 | 17 | — | |
YZDJQTHVDDOVHR
|
7.2 | Kd | 23 | — | |
OMIQRSKHABIPRH
|
7.2 | IC50 | 15 | — | |
UEJXELMBDCXXAQ
|
7.2 | IC50 | 9 | — | |
LAUHLGUSVSJYCI
|
7.2 | IC50 | 16 | — | |
JOOXLOJCABQBSG
|
7.1 | Kd | 139 | — | |
TXGKRVFSSHPBAJ
|
7.1 | IC50 | 11 | — | |
YZNIHXUBUWEUCM
|
7.0 | IC50 | 14 | — | |
NXSJMRCTGYTSTK
|
7.0 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
6.9 | Kd | 170 | — |