Target Details
| UniProt AC | P09668 |
|---|---|
| Gene Symbol | CTSH |
| Protein Name | Pro-cathepsin H |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 19
- Clinical molecules 1
- Avg pChEMBL 7.02
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (19)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YCYQOGPWUSMXGX
|
9.3 | Ki | 4 | — | |
YWXWRCMYHIYBSJ
|
8.8 | Ki | 4 | — | |
ZLZXUNHJWVLGTE
|
7.7 | IC50 | 4 | — | |
BEMWXCUECCHZDO
|
7.4 | IC50 | 4 | — | |
WNKGMQLRHKONID
|
7.4 | IC50 | 4 | — | |
DRRLOKQBVIVNIT
|
7.0 | IC50 | 5 | — | |
SZYYBVWPURUFRR
|
6.9 | IC50 | 8 | — | |
GLJZTHKUTGOBFU
|
6.9 | Ki | 4 | — | |
DVJGXMUWYFGXAS
|
6.8 | IC50 | 4 | Yes | |
LTLYEAJONXGNFG
|
6.7 | IC50 | 9 | — | |
VHDAHAMWVNXMSP
|
6.7 | IC50 | 7 | — | |
ZQXYZTRTLGOBEJ
|
6.7 | IC50 | 4 | — | |
ZQXYZTRTLGOBEJ
|
6.7 | IC50 | 4 | — | |
VUVLQWZOUOAKHY
|
6.6 | IC50 | 4 | — | |
VUVLQWZOUOAKHY
|
6.6 | IC50 | 4 | — | |
OLIMBXKACVCIMM
|
6.2 | IC50 | 3 | — | |
OLIMBXKACVCIMM
|
6.2 | IC50 | 3 | — | |
ITTAWEBSDKYKKK
|
6.2 | IC50 | 4 | — | |
VLZYXSQGILGQAI
|
6.2 | IC50 | 6 | — |