Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WLKXIKZJXFFRFT
|
8.2 | IC50 | 2 | — | |
YRUDYNCGPZHXRB
|
8.2 | Kd | 6 | — | |
DIMLYBUSJYNUFT
|
8.1 | Kd | 6 | — | |
FEWAGHIBDBSVCS
|
8.1 | IC50 | 2 | — | |
UHMOJOLDOBNIHB
|
8.1 | Ki | 6 | — | |
WGRLOIOBISATRO
|
8.1 | IC50 | 3 | — | |
ZUCUJAOPBDUFMB
|
8.1 | Ki | 6 | — | |
GCVSOKZESRXLDF
|
8.1 | IC50 | 2 | — | |
OFTYCXRAQKFFEW
|
8.1 | Ki | 6 | — | |
OUHRROUUMISCGY
|
8.1 | IC50 | 2 | — | |
DMWKBGXCJHQPFR
|
8.1 | IC50 | 2 | — | |
HESUKNSDMPJYHF
|
8.1 | Ki | 6 | — | |
JVYAUAVDPCSSTA
|
8.1 | IC50 | 2 | — | |
NXQOLSZAEQSUKO
|
8.1 | IC50 | 3 | — | |
ZZGOGKOPTVVJLD
|
8.1 | Ki | 6 | — | |
AISWQGLURAAAKE
|
8.1 | IC50 | 7 | — | |
CVWXJKQAOSCOAB
|
8.1 | Kd | 35 | — | |
OFMPMUCMGYQBDB
|
8.1 | IC50 | 2 | — | |
SDVCOWGIPMODEC
|
8.1 | IC50 | 18 | — | |
ABLAJTWOWSSMFU
|
8.1 | IC50 | 3 | — | |
CPMDPSXJELVGJG
|
8.1 | Ki | 6 | — | |
FFCFHBVSGILIJY
|
8.1 | Ki | 17 | — | |
GWVUCXTYNJIWGK
|
8.1 | Kd | 3 | — | |
HUMKYTSWTIZLSI
|
8.1 | Ki | 6 | — | |
JFJXNCYWRQBYGK
|
8.1 | Ki | 6 | — | |
MQLQJDVZLXXXAP
|
8.1 | Ki | 6 | — | |
SLOPYNWTLHFNFR
|
8.1 | IC50 | 2 | — | |
UDIUFPPEHOBBAN
|
8.1 | Ki | 6 | — | |
UFSGCADQVRKELP
|
8.1 | IC50 | 3 | — | |
VSVWQTDDGQSGHP
|
8.1 | Ki | 51 | — | |
WINHZLLDWRZWRT
|
8.1 | IC50 | 201 | Yes | |
WUWVRXPSSGTMJL
|
8.1 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
8.1 | IC50 | 165 | Yes | |
ZDEYUKODQZFZIK
|
8.1 | IC50 | 3 | — | |
ZKKRNZFCHLYOFH
|
8.1 | IC50 | 2 | — | |
ZWEHYQSGMOUIRZ
|
8.1 | IC50 | 3 | — | |
LFKPJUFFMOTFRX
|
8.1 | IC50 | 6 | — | |
MHITTXFPZXWLMH
|
8.1 | Kd | 6 | — | |
ODPGGGTTYSGTGO
|
8.1 | Kd | 153 | — | |
OINWQMFPLYPJMF
|
8.1 | IC50 | 3 | — | |
WJRBHBFXWWGLBI
|
8.1 | Ki | 6 | — | |
HWZNBJUXOVHGSL
|
8.1 | Ki | 6 | — | |
WJEOLQLKVOPQFV
|
8.1 | Kd | 24 | — | |
ZSWBFDGBEZTJRY
|
8.1 | IC50 | 4 | — | |
HUUDJQMFKCICDV
|
8.1 | Ki | 6 | — | |
PAHAOYHAOLZULX
|
8.1 | Ki | 6 | — | |
QCKVLRNZROXNAA
|
8.1 | IC50 | 2 | — | |
SDYGMEWQBSWSIW
|
8.1 | Kd | 6 | — | |
BLYDOULCQABGHT
|
8.1 | Ki | 6 | — | |
FJSAESWYZCNLQU
|
8.1 | Ki | 6 | — |