Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UZIDEIUGOKODKT
|
8.3 | IC50 | 2 | — | |
IFFBOVLYGJAFKB
|
8.3 | IC50 | 5 | — | |
MPYUMMWCLQVMLG
|
8.3 | IC50 | 11 | — | |
ZEHCAKZLQFXHKS
|
8.3 | IC50 | 2 | — | |
NGKALCMOLVCFHL
|
8.2 | Kd | 5 | — | |
SNHCRNMVYDHVDT
|
8.2 | IC50 | 3 | — | |
ZMZPKKALGYPJJM
|
8.2 | IC50 | 2 | — | |
BEIAIBOGYLFZCK
|
8.2 | IC50 | 4 | — | |
HUXJROJTQQSFPL
|
8.2 | IC50 | 2 | — | |
KGSOVEPCGRSZLN
|
8.2 | IC50 | 2 | — | |
SIUNALDMRGZQBR
|
8.2 | IC50 | 3 | — | |
VDGRPZZCHVECAN
|
8.2 | IC50 | 2 | — | |
XBUZLFQDBPBWCK
|
8.2 | Ki | 6 | — | |
XMTTXADILXOCTI
|
8.2 | IC50 | 2 | — | |
NCDVMWSJHOBWBM
|
8.2 | IC50 | 3 | — | |
UYWCBKUMESQOKL
|
8.2 | IC50 | 5 | — | |
HGJSLQXBCKJGHL
|
8.2 | IC50 | 2 | — | |
ITLNVPRPOQCABR
|
8.2 | IC50 | 2 | — | |
MPZNWDCJFYRKFH
|
8.2 | IC50 | 2 | — | |
NZUICIGFUCOURS
|
8.2 | IC50 | 4 | — | |
ODFKDTMBDLHPKM
|
8.2 | IC50 | 2 | — | |
UDLYZSYBPOFSSA
|
8.2 | IC50 | 2 | — | |
YEDBBOGEZDFFBL
|
8.2 | IC50 | 2 | — | |
YJSFAHMGDRBZGH
|
8.2 | IC50 | 16 | Yes | |
YKRJUNOOAMJFCU
|
8.2 | IC50 | 2 | — | |
CDOQYTRVCWQMJM
|
8.2 | Ki | 6 | — | |
GAKOWURXFQKQGU
|
8.2 | IC50 | 2 | — | |
MAWWXEIKARIPSX
|
8.2 | IC50 | 2 | — | |
IOXCZKDMVMERGD
|
8.2 | Ki | 6 | — | |
VHIADSOUXPEWOM
|
8.2 | Ki | 6 | — | |
WKQQROGAGZDSBZ
|
8.2 | Ki | 6 | — | |
FMCLDFJJIAZKCA
|
8.2 | Kd | 5 | — | |
JCKMPGSSOFUEAB
|
8.2 | IC50 | 2 | — | |
LHKUVOGMYOGQMG
|
8.2 | Ki | 6 | — | |
PRXJBBOPXMGUAC
|
8.2 | Ki | 6 | — | |
UKGLXBBBCMZJSW
|
8.2 | Ki | 6 | — | |
AAGVXWXEAOHUAD
|
8.2 | IC50 | 2 | — | |
AYBLFKIMJMUPEC
|
8.2 | Ki | 6 | — | |
BLNFXBVDIFFNQY
|
8.2 | IC50 | 2 | — | |
FUZNPGXZBNWJNB
|
8.2 | IC50 | 2 | — | |
HTYLSAJYCQVPBD
|
8.2 | IC50 | 3 | — | |
OIUSMJPCEZOFLD
|
8.2 | IC50 | 2 | — | |
OPRRAWCDBYHFFP
|
8.2 | IC50 | 3 | — | |
ORRNXRYWGDUDOG
|
8.2 | IC50 | 5 | — | |
PUHMCRONAFLMFJ
|
8.2 | IC50 | 2 | — | |
RFDYTLIVFMVNFI
|
8.2 | IC50 | 2 | — | |
STYDJMQKMJBSLF
|
8.2 | IC50 | 3 | — | |
TTYGGHQORNSTIY
|
8.2 | Ki | 6 | — | |
VCWSLEWLUZQPBS
|
8.2 | IC50 | 2 | — | |
WKHDSXVHKWSTGS
|
8.2 | IC50 | 2 | — |