Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZDNURMVOKAERHZ
|
8.4 | IC50 | 7 | Yes | |
ZQKNIPQNEVNCDY
|
8.4 | IC50 | 8 | — | |
GJWFUGSRILNJBR
|
8.4 | IC50 | 4 | — | |
KIVHIZZKZIPROE
|
8.4 | IC50 | 2 | — | |
VIWRJNDQSYSCMQ
|
8.4 | IC50 | 2 | — | |
YOZUNJXPGMAPQP
|
8.4 | IC50 | 2 | — | |
MMOPWANWYHZHPG
|
8.3 | IC50 | 3 | — | |
BYSPSKYBWHPEJW
|
8.3 | IC50 | 6 | — | |
FLYHUTANLWWHSP
|
8.3 | IC50 | 2 | — | |
GONLMECPQWNPOT
|
8.3 | IC50 | 2 | — | |
QFHBSJJMTUPRMF
|
8.3 | IC50 | 2 | — | |
ULHLSSWDQFLSBL
|
8.3 | IC50 | 6 | — | |
GARSAKHZBKMJHG
|
8.3 | IC50 | 2 | — | |
IONVXRPWTRMITM
|
8.3 | Ki | 6 | — | |
KWVDRTIIZKGPOQ
|
8.3 | Ki | 6 | — | |
PWULXWUQKORKGJ
|
8.3 | IC50 | 2 | — | |
YRQFTXBTINKLCO
|
8.3 | IC50 | 2 | — | |
ZASMEEJOVACSTK
|
8.3 | Ki | 6 | — | |
PIKYCWIZICBHRG
|
8.3 | Ki | 6 | — | |
PZYXWWIFXMVKBF
|
8.3 | IC50 | 2 | — | |
RHZNEYIWEJCIRC
|
8.3 | IC50 | 2 | — | |
ACCSYFAQPQXJJO
|
8.3 | Ki | 6 | — | |
CBPRXMDBGJCNJA
|
8.3 | IC50 | 2 | — | |
GGBRKXPKWAKIAS
|
8.3 | IC50 | 3 | — | |
GRDPLDYSIKQSRC
|
8.3 | IC50 | 3 | — | |
IFPFJZIFITZNRW
|
8.3 | IC50 | 2 | — | |
IVURVTQZRJNNOE
|
8.3 | IC50 | 4 | Yes | |
JMVVTEATJVVTPU
|
8.3 | Ki | 6 | — | |
JZGWDENJLOXKLZ
|
8.3 | IC50 | 4 | — | |
KSELTIXXASIVDL
|
8.3 | IC50 | 2 | — | |
MUWXXFVRGSATHH
|
8.3 | IC50 | 2 | — | |
MVKVCQNFFRDQDJ
|
8.3 | IC50 | 3 | — | |
NKEAAKWHNZZTLF
|
8.3 | IC50 | 2 | — | |
NQVBNOPSVRCGSI
|
8.3 | IC50 | 2 | — | |
OEZUXIBNCYTQAV
|
8.3 | IC50 | 5 | Yes | |
QAQWRVQXBRITDM
|
8.3 | IC50 | 4 | — | |
QLGPUCHJSSSJAW
|
8.3 | IC50 | 2 | — | |
RIVKJCNOYQAWOL
|
8.3 | IC50 | 3 | — | |
SHKVYTQIJOOEMA
|
8.3 | IC50 | 6 | — | |
XXJWYDDUDKYVKI
|
8.3 | Kd | 52 | — | |
YIQKRGSTCNRKES
|
8.3 | Ki | 6 | — | |
YXZQRTLGEGYVTJ
|
8.3 | IC50 | 2 | — | |
COYNQUUUEZTJFP
|
8.3 | IC50 | 2 | — | |
CTRSFSGBUZZONS
|
8.3 | IC50 | 2 | — | |
PMNKHDAXQLPDIQ
|
8.3 | IC50 | 2 | — | |
BEBIBSIUUZHXBI
|
8.3 | IC50 | 3 | — | |
JXZTVKIJNMZSJO
|
8.3 | IC50 | 2 | — | |
KGSFRFBLOVIBMQ
|
8.3 | IC50 | 2 | — | |
QOVBTXBRBQUBBP
|
8.3 | IC50 | 3 | — | |
NYKOXJAXPORIHO
|
8.3 | Ki | 6 | — |