Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OBFGRWOUNPRHNH
|
8.5 | IC50 | 6 | — | |
YYHLHURAZWXOQD
|
8.5 | IC50 | 2 | — | |
KYABXXGGLXXKNT
|
8.5 | IC50 | 2 | — | |
LFYIJZIUOBYEBW
|
8.5 | IC50 | 2 | — | |
FGDPUUPSGZJLCV
|
8.5 | IC50 | 2 | — | |
IOELWNQBJITVMV
|
8.5 | IC50 | 2 | — | |
QOSFVUGBELGFPJ
|
8.5 | IC50 | 2 | — | |
TZSBMAHRPWFGJQ
|
8.5 | IC50 | 2 | — | |
VKXQKNIMTYWKSX
|
8.5 | IC50 | 2 | — | |
YVIQBACAFGCINI
|
8.5 | IC50 | 2 | — | |
AZWGTRFPZWYXCN
|
8.4 | IC50 | 2 | — | |
GLLDYCCWAIPJAY
|
8.4 | IC50 | 2 | — | |
TWWKXZDIDHDHRF
|
8.4 | IC50 | 7 | — | |
WYFQWNLCVLJDGA
|
8.4 | IC50 | 2 | — | |
YCQZVDKPIKTXSN
|
8.4 | IC50 | 2 | — | |
DSYCVJBNOBWEDH
|
8.4 | IC50 | 2 | — | |
HLUJJJCUMAOJIP
|
8.4 | IC50 | 2 | — | |
QOPDGZWWDPNCDK
|
8.4 | IC50 | 2 | — | |
SSMFYNNDUCDQGD
|
8.4 | IC50 | 2 | — | |
CPKWNMKGJMCCPZ
|
8.4 | IC50 | 2 | — | |
GBFDLYAUGOZCIP
|
8.4 | IC50 | 2 | — | |
JRWQMURFOYPHJJ
|
8.4 | IC50 | 2 | — | |
LZQMVZQCOPEYQN
|
8.4 | IC50 | 2 | — | |
YVNXWNFAWUVVND
|
8.4 | IC50 | 2 | — | |
JHWZPTAZWZKCEQ
|
8.4 | IC50 | 5 | — | |
KEFBHUKKKFYQSI
|
8.4 | IC50 | 2 | — | |
LMCLMMAYWZRBRH
|
8.4 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
8.4 | Kd | 137 | Yes | |
XKKWYUUBWNYGNI
|
8.4 | IC50 | 2 | — | |
ZXYVWKYLUPYZGL
|
8.4 | Kd | 5 | — | |
QOPDGZWWDPNCDK
|
8.4 | IC50 | 2 | — | |
XVMRGPVSAKTURK
|
8.4 | IC50 | 2 | — | |
DBDUMMKYYKJJID
|
8.4 | IC50 | 3 | — | |
GFHOQPFRWWTZIG
|
8.4 | IC50 | 2 | — | |
GKEYKDOLBLYGRB
|
8.4 | IC50 | 3 | — | |
HWXPNIATGYCXGR
|
8.4 | IC50 | 2 | — | |
KVRUUDPIAWUBGE
|
8.4 | IC50 | 2 | — | |
LMEJZAGBGSRBJA
|
8.4 | IC50 | 2 | — | |
LYWLFOKRWJGIJX
|
8.4 | IC50 | 3 | — | |
OICXIBPVOXVRBW
|
8.4 | IC50 | 4 | Yes | |
OVKRRHLOFQLWRN
|
8.4 | IC50 | 2 | — | |
OVTHZKRCTBBAOW
|
8.4 | IC50 | 5 | Yes | |
PCPXTLXXRRQODN
|
8.4 | IC50 | 2 | — | |
QJOMTUGNMKUBCP
|
8.4 | IC50 | 3 | — | |
TWYCZJMOEMMCGC
|
8.4 | IC50 | 6 | Yes | |
WDDLXDTWOAENKE
|
8.4 | IC50 | 5 | Yes | |
YYPVGQBXTJNGFW
|
8.4 | IC50 | 4 | — | |
HZHDGZNDKAIYRX
|
8.4 | IC50 | 2 | — | |
WYGBVKGNAJVGTR
|
8.4 | IC50 | 2 | — | |
XHPCNYYPHRXXOG
|
8.4 | IC50 | 2 | — |