Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DZSUJUOJJJCWGG
|
8.6 | IC50 | 55 | Yes | |
JVKHSWZCCXPYQY
|
8.6 | IC50 | 2 | — | |
RZJJNSILMXCYNX
|
8.6 | IC50 | 2 | — | |
XBNLLMKPDMJSKX
|
8.6 | IC50 | 2 | — | |
INOASWZOZPQAQM
|
8.6 | Kd | 5 | — | |
BGVQPQHIUOTLBT
|
8.6 | Kd | 6 | — | |
LVMAULGVWBINFP
|
8.6 | IC50 | 6 | — | |
SUXYGJZMCWKJJI
|
8.6 | IC50 | 26 | Yes | |
HKSZLNNOFSGOKW
|
8.6 | IC50 | 408 | — | |
HTJGFHHVVPNDMR
|
8.6 | IC50 | 6 | — | |
ZMLDVKWBDWLLML
|
8.6 | IC50 | 2 | — | |
LRVCIMMMXCELJH
|
8.6 | IC50 | 2 | — | |
UVRLRMVYKSBGHX
|
8.6 | IC50 | 2 | — | |
VAWLAPYBUJTXRS
|
8.6 | IC50 | 6 | Yes | |
FRYZXBGRKYRYQL
|
8.5 | IC50 | 2 | — | |
HEJZALDKCWDYLL
|
8.5 | IC50 | 2 | — | |
OHRPYVMGIKIEMB
|
8.5 | IC50 | 2 | — | |
PVZJLPGZMRIHCQ
|
8.5 | IC50 | 3 | — | |
RCZHVXSTTOXWRM
|
8.5 | IC50 | 3 | — | |
YXXHOBHYIQNGNP
|
8.5 | IC50 | 2 | — | |
KNBUIVITEDSJDJ
|
8.5 | IC50 | 2 | — | |
KRFPEYFNZCXMCV
|
8.5 | IC50 | 2 | — | |
UHRAUSTWOGDPJJ
|
8.5 | IC50 | 2 | — | |
BJTVHTAPKJNNGR
|
8.5 | IC50 | 3 | — | |
CZSOWVHBIBQBJU
|
8.5 | IC50 | 2 | — | |
DEEVAXGZAJDWSB
|
8.5 | IC50 | 2 | — | |
DPRXHQKZIFLCDL
|
8.5 | IC50 | 2 | — | |
DYSDUQPAIATDAA
|
8.5 | IC50 | 5 | Yes | |
GSURAMUGDNSWKE
|
8.5 | IC50 | 3 | — | |
HPPAKEIARRFUBB
|
8.5 | IC50 | 4 | — | |
KPVSGWFUYLJRIW
|
8.5 | IC50 | 2 | — | |
KVZJZSJXYMDYPE
|
8.5 | IC50 | 2 | — | |
LQNNUQKZSZVOBC
|
8.5 | IC50 | 2 | — | |
NSTFTWHSPRGGFB
|
8.5 | IC50 | 2 | — | |
OSEYUXXMDLYZKE
|
8.5 | IC50 | 5 | Yes | |
QILQUYGQJMWOFT
|
8.5 | IC50 | 3 | Yes | |
RWBSHLPMAISSHT
|
8.5 | IC50 | 3 | — | |
WPHKIQPVPYJNAX
|
8.5 | IC50 | 81 | — | |
XDDLRMCIDZLHNL
|
8.5 | IC50 | 3 | — | |
XPLJEFSRINKZLC
|
8.5 | IC50 | 5 | Yes | |
NXTAONONNMIHOO
|
8.5 | IC50 | 3 | — | |
YISMQBFJYDFMAL
|
8.5 | IC50 | 46 | — | |
NKEUPUJTVALZIK
|
8.5 | Ki | 28 | — | |
NWMPVMMGSHXANZ
|
8.5 | Ki | 58 | — | |
BWHGTIFBFVAAKP
|
8.5 | IC50 | 2 | — | |
GJWFUGSRILNJBR
|
8.5 | IC50 | 4 | — | |
KHKKHXIFTCUDNT
|
8.5 | IC50 | 2 | — | |
XJWRVUVWWHDVEF
|
8.5 | IC50 | 2 | — | |
FNBMUJLNNOOTMF
|
8.5 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
8.5 | Kd | 220 | — |