Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVGJYTZRLNHLDH
|
8.7 | IC50 | 2 | — | |
DGEKRKGWIXOURE
|
8.7 | IC50 | 2 | — | |
HQSVYZWDHYEPBY
|
8.7 | IC50 | 2 | — | |
YYPOHOIDTCSCHL
|
8.7 | IC50 | 2 | — | |
ZOKZHFIBKOVHBQ
|
8.7 | IC50 | 2 | — | |
HNAKAPUKEWMJOX
|
8.7 | IC50 | 2 | — | |
JYRPSPNQBJTHFR
|
8.7 | IC50 | 2 | — | |
NZUGNTZEMQTKDH
|
8.7 | IC50 | 2 | — | |
XSYZCQDIHCJKAQ
|
8.7 | IC50 | 2 | — | |
NZDHEVOTZDNDBN
|
8.7 | IC50 | 2 | — | |
SOBMUPLZQRAPEL
|
8.7 | IC50 | 2 | — | |
XTPMOIFZATWEBG
|
8.7 | IC50 | 2 | — | |
BWLBVHWCNZAPOW
|
8.7 | IC50 | 4 | — | |
BZAOYXZLPUIEJZ
|
8.7 | IC50 | 2 | — | |
CCIRQCXOVCNPBI
|
8.7 | IC50 | 3 | — | |
DKNUPRMJNUQNHR
|
8.7 | Kd | 33 | — | |
GJKVMXDBPDDFHI
|
8.7 | Ki | 27 | — | |
HGAQQKPBNGSIMU
|
8.7 | IC50 | 3 | Yes | |
JAAZVIPSQFETPP
|
8.7 | IC50 | 3 | — | |
JVYWSDGZGNKUKM
|
8.7 | IC50 | 3 | — | |
LUQXZVFBJJZMSL
|
8.7 | IC50 | 2 | — | |
NZTCZQRXCIAJMP
|
8.7 | IC50 | 5 | Yes | |
QPNALTDCQOTWLI
|
8.7 | IC50 | 4 | Yes | |
QZXMREJVHYOFOD
|
8.7 | IC50 | 2 | — | |
RDWQPGCGRCTSIN
|
8.7 | IC50 | 5 | Yes | |
SVEZALKOLCCBNB
|
8.7 | IC50 | 2 | — | |
UPDDTKQTXDTPHV
|
8.7 | IC50 | 2 | — | |
XLZFINWQTYEKJR
|
8.7 | IC50 | 5 | Yes | |
HZORURMFPRFGNI
|
8.7 | IC50 | 2 | — | |
JEZNQOLZSHORKU
|
8.7 | IC50 | 2 | — | |
JSUWTFPXDRARTH
|
8.7 | IC50 | 2 | — | |
FOKQTIHUENEYBC
|
8.7 | IC50 | 2 | — | |
HUQSQQXBXUUYED
|
8.7 | IC50 | 2 | — | |
NYBNNHFUSGTOBH
|
8.7 | IC50 | 2 | — | |
SGQQSWUDPWLSBL
|
8.7 | IC50 | 2 | — | |
UYLCGOHBKJOVLW
|
8.7 | IC50 | 2 | — | |
KYABXXGGLXXKNT
|
8.7 | IC50 | 2 | — | |
GCUZSJPHOPKZNQ
|
8.7 | IC50 | 2 | — | |
OEUMLQMTMOCCGW
|
8.7 | Kd | 6 | — | |
BBDMMLFJRXKDIR
|
8.7 | IC50 | 2 | — | |
RJOOYQPEJJZEIP
|
8.7 | IC50 | 2 | — | |
OIANGKGOYKDGQV
|
8.6 | Kd | 10 | — | |
QBRQTJMZEYORSP
|
8.6 | Kd | 12 | — | |
UQQZPUPMXFCRML
|
8.6 | IC50 | 4 | — | |
VPSOGOXLPQRTAD
|
8.6 | IC50 | 2 | — | |
XFGKIMCSRPXPMT
|
8.6 | IC50 | 2 | — | |
HXDDZHMPEAWUHJ
|
8.6 | IC50 | 2 | — | |
IMFSTVJNACYASP
|
8.6 | IC50 | 2 | — | |
YPLJOKYMNOWDIM
|
8.6 | IC50 | 2 | — | |
AAKYKCSHUIKMET
|
8.6 | IC50 | 2 | — |