Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NDZHXVIMTDMQGZ
|
9.1 | IC50 | 4 | — | |
WEZLSLVHHILOGK
|
9.1 | IC50 | 3 | — | |
XALOFLMEUAMOLD
|
9.1 | IC50 | 3 | — | |
LCFJBBWUVXKZGB
|
9.0 | IC50 | 2 | — | |
VDTIARDTOLLQLW
|
9.0 | IC50 | 2 | — | |
LFXRUSJBXAQXCD
|
9.0 | IC50 | 2 | — | |
NNYCTPRWKDDLFA
|
9.0 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
9.0 | Kd | 43 | — | |
SEJGTFPOEJWEGG
|
9.0 | Kd | 149 | — | |
IFOVLFYNYABOTP
|
9.0 | IC50 | 2 | — | |
CTUNMKNUSCLTQS
|
9.0 | IC50 | 2 | — | |
DIKCCHQBRVVDJR
|
9.0 | IC50 | 2 | Yes | |
JBIRTAVBFDUZQN
|
9.0 | IC50 | 2 | — | |
JQDTYPFSLIFJAT
|
9.0 | IC50 | 5 | Yes | |
JVCWPUFNLFSKFS
|
9.0 | Kd | 5 | — | |
LOCPAEPNEIAJSG
|
9.0 | IC50 | 2 | — | |
OQLVVMGCNQOROZ
|
9.0 | IC50 | 2 | — | |
QIZGCINCAAEMBX
|
9.0 | IC50 | 2 | — | |
ROHJEIACUNTGFP
|
9.0 | IC50 | 16 | — | |
SCUGTCMSRMQNNQ
|
9.0 | IC50 | 7 | — | |
SRSGVKWWVXWSJT
|
9.0 | IC50 | 3 | Yes | |
UMBIRSZUCJNBHB
|
9.0 | IC50 | 18 | — | |
VKBFHTIUXUCYRQ
|
9.0 | Ki | 66 | — | |
WINHZLLDWRZWRT
|
9.0 | Ki | 66 | — | |
WNVADWMUVOLRPY
|
9.0 | IC50 | 3 | — | |
WSBZFFNSBMBYQA
|
9.0 | IC50 | 9 | — | |
YCNDQMGBKRXDNQ
|
9.0 | IC50 | 3 | — | |
JQWRPCZUMWGJSB
|
9.0 | IC50 | 2 | — | |
QIZGCINCAAEMBX
|
9.0 | IC50 | 2 | — | |
QIZGCINCAAEMBX
|
9.0 | IC50 | 2 | — | |
RXZNKADVZBVZKL
|
9.0 | IC50 | 2 | — | |
BUZZYBLUNDCBEB
|
9.0 | IC50 | 2 | — | |
AQSSMEORRLJZLU
|
9.0 | IC50 | 34 | Yes | |
PAHBMDHIMGYJEW
|
9.0 | IC50 | 2 | — | |
JEZNQOLZSHORKU
|
8.9 | IC50 | 2 | — | |
XMFJUJPBMXFKQN
|
8.9 | IC50 | 2 | — | |
CTUNMKNUSCLTQS
|
8.9 | IC50 | 2 | — | |
VZDAKDOJJGVGBR
|
8.9 | IC50 | 2 | — | |
JUAOOEGSHIUSJA
|
8.9 | IC50 | 2 | — | |
DNLQIFRJOZJGCU
|
8.9 | IC50 | 6 | Yes | |
NGKALCMOLVCFHL
|
8.9 | Kd | 5 | — | |
PHXJVRSECIGDHY
|
8.9 | IC50 | 59 | — | |
REYMYGJJLFMJCU
|
8.9 | IC50 | 2 | — | |
DVHSIXNBKKXFCJ
|
8.9 | IC50 | 2 | — | |
QGTNBHVHNFUNSQ
|
8.9 | IC50 | 2 | — | |
UULYXELMKPCXOS
|
8.9 | IC50 | 2 | — | |
ADLPKFFMGIJZIM
|
8.9 | Ki | 44 | — | |
MRYVITFPRDXAHG
|
8.9 | IC50 | 2 | — | |
WYCNEMUMQDPFHP
|
8.9 | IC50 | 2 | — | |
ZMZGUJSLGMATGF
|
8.9 | IC50 | 5 | — |