Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SLWDPPUDEOJKMG
|
7.9 | IC50 | 2 | — | |
GWQQUSRBNJRKLG
|
7.9 | IC50 | 3 | — | |
JINRJKYXFRZRJB
|
7.9 | IC50 | 2 | — | |
LHZZZBFUJPHNCR
|
7.9 | Ki | 6 | — | |
VBCPAAMHSAMKFK
|
7.9 | Ki | 6 | — | |
WNMAXXDDBQOLPI
|
7.9 | IC50 | 5 | — | |
WNNZGWZQLJGBNE
|
7.9 | Ki | 6 | — | |
BMWHAGVKNLRXNW
|
7.9 | IC50 | 3 | — | |
DZFZXPPHBWCXPQ
|
7.9 | IC50 | 12 | — | |
KBUOUGKAAPDJRZ
|
7.9 | IC50 | 2 | — | |
LJFSJSPWQGPGIK
|
7.9 | Ki | 6 | — | |
LVHJAVYIDITWAZ
|
7.9 | IC50 | 2 | — | |
NAZMMUDKWQHGKI
|
7.9 | IC50 | 2 | — | |
NNBXSFREJXVASG
|
7.9 | IC50 | 2 | — | |
QLCHTTFSIBNNDD
|
7.9 | IC50 | 2 | — | |
REMWVXFHAPBPEU
|
7.9 | IC50 | 3 | — | |
SQMMWBVSXONNAM
|
7.9 | Ki | 6 | — | |
VBQLMMTYTIVERQ
|
7.9 | Ki | 6 | — | |
VLIWYQAUGIWSFX
|
7.9 | Ki | 6 | — | |
XESKGZXKYIRKRJ
|
7.9 | Ki | 6 | — | |
KSXXLYFDRDYXJK
|
7.9 | IC50 | 3 | — | |
WEWNFYSPKIFAFJ
|
7.9 | IC50 | 2 | — | |
ZNFMAXYFBGIDKY
|
7.9 | IC50 | 3 | — | |
VWWWKWXBDHJDSL
|
7.9 | IC50 | 2 | — | |
VZQHANSAAHZYGF
|
7.9 | IC50 | 2 | — | |
AOHLFNGYVXMGNP
|
7.8 | Ki | 6 | — | |
DFGKWRXDDUYBAT
|
7.8 | Ki | 6 | — | |
DGECBIQUJWBSOF
|
7.8 | IC50 | 3 | — | |
GUHBTJGSLWFLFC
|
7.8 | IC50 | 2 | — | |
HSKISFLIRPOYCF
|
7.8 | IC50 | 5 | — | |
KNXQEJUJQOZAKP
|
7.8 | IC50 | 7 | Yes | |
OLBVLPUBUBRBGW
|
7.8 | Ki | 6 | — | |
RUSCZKWQARTAPP
|
7.8 | IC50 | 3 | — | |
UEPXBTCUIIGYCY
|
7.8 | Kd | 6 | — | |
XALNEEALNAULMH
|
7.8 | IC50 | 3 | — | |
ZLUSJKSRLQNGJZ
|
7.8 | IC50 | 3 | — | |
ALKQTTOWJRBJBP
|
7.8 | IC50 | 2 | — | |
DGUYNPBHMTWHCX
|
7.8 | IC50 | 2 | — | |
LYBAWURNJUOHRS
|
7.8 | Ki | 6 | — | |
RQJCPYMTCVHMBN
|
7.8 | Ki | 6 | — | |
VPXYJYVAKTVLLA
|
7.8 | IC50 | 2 | — | |
ZDZUIAHQMAWKQF
|
7.8 | IC50 | 2 | — | |
GHHLGOSWKKKPAV
|
7.8 | IC50 | 2 | — | |
ACAVWBSORQCXCG
|
7.8 | IC50 | 2 | — | |
APPAUNZXIPSWAS
|
7.8 | IC50 | 7 | Yes | |
BRFOGQVFBWDQGX
|
7.8 | IC50 | 6 | — | |
DKFVXLBMKSCYMJ
|
7.8 | Ki | 6 | — | |
HTJCJGPUYPCIIH
|
7.8 | IC50 | 2 | — | |
JVGNHFZOVWJKER
|
7.8 | IC50 | 3 | — | |
OSHAGQCZZMYWEP
|
7.8 | IC50 | 3 | — |