Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SILANKVZJSUJHJ
|
8.0 | IC50 | 9 | — | |
SQUBJXXBYMPOFW
|
8.0 | IC50 | 6 | Yes | |
SZJRFGYYRZITCZ
|
8.0 | IC50 | 4 | — | |
UIQHNAPAGAHZFT
|
8.0 | IC50 | 2 | — | |
UNYBBLITYOSZKC
|
8.0 | IC50 | 2 | — | |
VMNBDLPXPRVHFM
|
8.0 | Ki | 6 | — | |
WIICWOVXHJZGNO
|
8.0 | IC50 | 2 | — | |
WWSUCZQRKHASNA
|
8.0 | IC50 | 3 | — | |
XNOHHMMIXCDTFE
|
8.0 | Ki | 6 | — | |
YVNKPHLJKPWZRT
|
8.0 | IC50 | 4 | — | |
KILPAWAZPJHBFA
|
8.0 | Ki | 6 | — | |
PGQJZWZFOOWFNP
|
8.0 | Ki | 6 | — | |
SCCKBJZRORUBHR
|
8.0 | Ki | 6 | — | |
YYICSPRZBVQPTF
|
8.0 | Ki | 6 | — | |
ASUVAFYTTOHJIF
|
8.0 | IC50 | 2 | — | |
DLUVOPPDOKCLLX
|
8.0 | IC50 | 2 | — | |
QUTYYJGQIXIMSJ
|
8.0 | Ki | 6 | — | |
RJIWXRGRXHMIJN
|
8.0 | Ki | 6 | — | |
VTBJZDMBUWEQBI
|
8.0 | IC50 | 2 | — | |
DQGTWWTUKZRUKI
|
8.0 | IC50 | 3 | — | |
JJLJYAPQIYLGFI
|
8.0 | Ki | 6 | — | |
LFNAERHMPRGPKC
|
8.0 | IC50 | 2 | — | |
MCTXSDCWFQAGFS
|
8.0 | IC50 | 3 | — | |
OMWAXUAYDHMCSG
|
8.0 | Ki | 6 | — | |
PETRONSJSNBTST
|
8.0 | Ki | 6 | — | |
RCMWTMHAMLWFGA
|
8.0 | Ki | 6 | — | |
UBICMXXPSIFNBD
|
8.0 | IC50 | 2 | — | |
VPWJHKVHKZOWKO
|
8.0 | Ki | 6 | — | |
WJXCYXYVNGMHAO
|
8.0 | IC50 | 2 | — | |
OSKVLQNSYZYKLO
|
8.0 | Ki | 6 | — | |
VLIWYQAUGIWSFX
|
8.0 | Ki | 6 | — | |
ZOTWWNJHIZTSQU
|
8.0 | IC50 | 2 | — | |
AVRHXSYMJIZSHR
|
7.9 | Ki | 6 | — | |
BCAHGWFHBBMPHP
|
7.9 | IC50 | 2 | — | |
MMKGCMKHOQBTJH
|
7.9 | Ki | 6 | — | |
RDKKLWLGQWWMHQ
|
7.9 | Ki | 6 | — | |
CPLREIYJOXSORV
|
7.9 | Ki | 6 | — | |
DPKYVXPTKBMCDY
|
7.9 | Ki | 6 | — | |
AAKJLRGGTJKAMG
|
7.9 | IC50 | 50 | Yes | |
FCLMAXRVUCVWGI
|
7.9 | IC50 | 2 | — | |
HHPVWJJNJSJOLQ
|
7.9 | IC50 | 3 | — | |
KESUAIOCJKBPRI
|
7.9 | IC50 | 3 | — | |
PETGNDYNMCNUKJ
|
7.9 | IC50 | 3 | — | |
QTAROSPVYXDUDL
|
7.9 | IC50 | 2 | — | |
RCHBURXYVZCGRM
|
7.9 | IC50 | 2 | — | |
RKESDYSOJBSAAE
|
7.9 | IC50 | 3 | — | |
SZPKERXOPUWUPW
|
7.9 | IC50 | 3 | — | |
UVZUIESPIIIPQW
|
7.9 | IC50 | 3 | — | |
WVOFZQPJICMMLE
|
7.9 | IC50 | 3 | — | |
DHONEALZRPCJOV
|
7.9 | Ki | 6 | — |