Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPIULPPERVHOJE
|
8.1 | IC50 | 2 | — | |
WJTZIBDSNXVBCN
|
8.1 | Ki | 6 | — | |
BHBBGXQSTGBYSZ
|
8.1 | IC50 | 2 | — | |
CAAQXWCBWGARSL
|
8.1 | IC50 | 3 | — | |
FVVWICPRPMXEEL
|
8.1 | IC50 | 2 | — | |
KXLRYMPSHOVNJE
|
8.1 | IC50 | 6 | — | |
SDQXQGSVVDEHLF
|
8.1 | IC50 | 2 | — | |
SSSVBCHLFDKMBI
|
8.1 | Ki | 6 | — | |
UZYXETLFKQALDE
|
8.1 | IC50 | 3 | — | |
YQVZJSYFTHDUNC
|
8.1 | IC50 | 2 | — | |
GUQSJGOTOKVEDW
|
8.0 | IC50 | 2 | — | |
LTJCRCKPWKQPOV
|
8.0 | Ki | 6 | — | |
RAHBGWKEPAQNFF
|
8.0 | Kd | 26 | — | |
DYHVAHJSHIYCLL
|
8.0 | IC50 | 4 | — | |
JLFPGEKGHMUMDY
|
8.0 | Ki | 6 | — | |
KIRQJJFAFLYYJQ
|
8.0 | Ki | 6 | — | |
WDUSDNGPVZEHRQ
|
8.0 | Ki | 6 | — | |
YNFGJAAJMZXYQP
|
8.0 | Ki | 6 | — | |
ZTLIJXDSHRPKGC
|
8.0 | IC50 | 2 | — | |
BCVBGCRLWBQIAF
|
8.0 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
8.0 | IC50 | 154 | — | |
FHTTVJXLZSYAJH
|
8.0 | Ki | 6 | — | |
MKBJXBMPLSSNMX
|
8.0 | Ki | 6 | — | |
QLGQYEDJCJVGFI
|
8.0 | Ki | 6 | — | |
TTXOTMLADFPMGH
|
8.0 | IC50 | 2 | — | |
YTHUQGIGAIZNIM
|
8.0 | IC50 | 3 | — | |
ZBQPGWRCYGZRMB
|
8.0 | Ki | 6 | — | |
WUEKYNCXBMROQI
|
8.0 | Ki | 6 | — | |
APYYTEJNOZQZNA
|
8.0 | IC50 | 3 | Yes | |
AYXVSCVVQIADBF
|
8.0 | Ki | 10 | — | |
BZZIQPCXCNKABW
|
8.0 | IC50 | 2 | Yes | |
CFAOCANWUGXOIL
|
8.0 | Ki | 6 | — | |
CNIWCJQSFDYIDI
|
8.0 | IC50 | 3 | — | |
DIWNHTDZEZGKJK
|
8.0 | IC50 | 3 | — | |
DRGIYHQKZKDPLX
|
8.0 | IC50 | 2 | — | |
FNVHVYCXTFAQSG
|
8.0 | Ki | 6 | — | |
FPYCSQMCBIGNHK
|
8.0 | IC50 | 3 | — | |
FWRUVEHMIVRQGU
|
8.0 | IC50 | 2 | — | |
FZMROVZIFREMDI
|
8.0 | IC50 | 2 | — | |
GBLFVKOVMVPIQF
|
8.0 | IC50 | 2 | — | |
GCKTWBJEXJWFHY
|
8.0 | IC50 | 18 | — | |
JWITUUPNOFPOGN
|
8.0 | IC50 | 3 | — | |
JZKVGXOGXXCAKW
|
8.0 | IC50 | 3 | — | |
KGSRYTUWXUESJK
|
8.0 | IC50 | 7 | — | |
LJZDAUHIEXUPMS
|
8.0 | IC50 | 4 | — | |
LUIRMPBUMLMGFN
|
8.0 | IC50 | 2 | — | |
NECQZMQPXFYVOY
|
8.0 | Ki | 26 | — | |
NGBFROQDGZCMCE
|
8.0 | IC50 | 3 | — | |
NXFMFUNSRYFXMH
|
8.0 | Ki | 6 | — | |
OOQTVBOFLACKQI
|
8.0 | IC50 | 2 | — |