Target Details
| UniProt AC | P09619 |
|---|---|
| Gene Symbol | PDGFRB |
| Protein Name | Platelet-derived growth factor receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF13927 (Ig_3) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,527
- Clinical molecules 200
- Avg pChEMBL 7.52
KEGG Pathways (21)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Focal adhesion
- Gap junction
- Glioma
- Human papillomavirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (6)
Active Molecules (1,527)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCCPLJOKGAACRT
|
10.1 | Kd | 599 | — | |
CTUHJNJXPMROFF
|
10.0 | IC50 | 3 | — | |
ZJQHYAYIOMPFGN
|
10.0 | IC50 | 3 | — | |
NNFDRCGXLJTASH
|
9.8 | IC50 | 4 | — | |
CLNJNVQBKCEOLA
|
9.7 | IC50 | 3 | — | |
SDLZNEBGHGGFNW
|
9.7 | IC50 | 3 | — | |
TVMVUMUJXVSING
|
9.7 | IC50 | 3 | Yes | |
CTNPALGJUAXMMC
|
9.5 | Kd | 151 | — | |
SHPFDGWALWEPGS
|
9.5 | Kd | 35 | — | |
BBEVMAFPVMSMEU
|
9.5 | IC50 | 3 | — | |
HWEVEQFMAGTKGM
|
9.5 | IC50 | 3 | — | |
OZIZBAWFMYRHDD
|
9.5 | IC50 | 3 | — | |
VPDYUDURNXPNMA
|
9.5 | IC50 | 5 | Yes | |
KUNZDWIFPOMUOX
|
9.5 | Ki | 36 | — | |
KTZAHPAGCSCZTG
|
9.4 | IC50 | 3 | — | |
MMCWBZCSGNCOMQ
|
9.4 | IC50 | 5 | Yes | |
RTYJMUXLFRYRBU
|
9.4 | Ki | 35 | — | |
SXAVOOSGLYHVJW
|
9.4 | IC50 | 4 | — | |
XLYVQVWMTOLDNL
|
9.4 | IC50 | 21 | — | |
XLYVQVWMTOLDNL
|
9.4 | IC50 | 21 | — | |
JPJAUHSLJCUGAH
|
9.4 | IC50 | 4 | — | |
WRVJJQONQSKWPP
|
9.4 | IC50 | 2 | — | |
PPUIQOGYMIRZOS
|
9.3 | IC50 | 2 | — | |
HOOKXRVARVUTOQ
|
9.3 | IC50 | 2 | — | |
BRTHUECZMVKNMQ
|
9.3 | Ki | 31 | — | |
MBTDIENWIYANIG
|
9.3 | IC50 | 5 | Yes | |
MDNAJFVDTSUEGN
|
9.3 | IC50 | 3 | — | |
OFGUFFNSCXNTNV
|
9.3 | IC50 | 4 | — | |
PWPWTOPEJWNZOA
|
9.2 | IC50 | 3 | — | |
APJYLVNVUZIPJQ
|
9.2 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
9.2 | Ki | 33 | — | |
ZBNZXTGUTAYRHI
|
9.2 | Kd | 102 | Yes | |
JVVXCTKZKBXESA
|
9.2 | IC50 | 2 | — | |
INFXGMKRYCEOFJ
|
9.2 | IC50 | 4 | — | |
JJNUVTXMRDPOPO
|
9.2 | IC50 | 3 | — | |
BGIYONAQBFCOPI
|
9.1 | IC50 | 2 | — | |
OPTZTHAQEZWUIM
|
9.1 | IC50 | 2 | — | |
WJIAKJKQRZFXIW
|
9.1 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
9.1 | Ki | 118 | — | |
JGFZPZGREYNUPH
|
9.1 | IC50 | 5 | Yes | |
JRHZSLDMBCJCRQ
|
9.1 | IC50 | 2 | — | |
VCFDMLBPASGZTP
|
9.1 | Ki | 38 | — | |
AQGHUQFARNGYDN
|
9.1 | IC50 | 2 | — | |
NGKALCMOLVCFHL
|
9.1 | Kd | 5 | — | |
SIFWORLXBPDHFA
|
9.1 | IC50 | 2 | — | |
QSMHVQQDSGOSQI
|
9.1 | IC50 | 2 | — | |
ZIVQDWVIGMBANJ
|
9.1 | IC50 | 2 | — | |
KXENZBKDXGJGBN
|
9.1 | IC50 | 2 | — | |
VLTUYLMKVNYVHY
|
9.1 | IC50 | 2 | — | |
BFZLDRFGXXMKES
|
9.1 | IC50 | 5 | Yes |