Target Details
| UniProt AC | P09238 |
|---|---|
| Gene Symbol | MMP10 |
| Protein Name | Stromelysin-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 133
- Clinical molecules 5
- Avg pChEMBL 6.99
Active Molecules (133)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SJWYFGLDVUQIEF
|
6.4 | Ki | 4 | — | |
VCJGVCZITQVJET
|
6.4 | Ki | 4 | — | |
AEOWLQGPNGMHBP
|
6.3 | Ki | 8 | — | |
BVKYTKVUMKYONQ
|
6.3 | Ki | 5 | — | |
RDMHVXDIUPIFCJ
|
6.3 | IC50 | 4 | — | |
YXSJVSGLVWXWOT
|
6.3 | IC50 | 4 | — | |
LWAJTROMLACBIU
|
6.3 | IC50 | 2 | — | |
BJBJSCJDKGVTKQ
|
6.3 | IC50 | 2 | — | |
QQGKYSPTORHWNZ
|
6.3 | Ki | 6 | — | |
MFTZEUCXFCXINH
|
6.3 | Ki | 6 | — | |
NZUPMMOEPOVBQE
|
6.3 | Ki | 5 | — | |
PNAVYQLZJZNXTL
|
6.3 | IC50 | 2 | — | |
WNEMBEALMHVXIK
|
6.3 | IC50 | 7 | — | |
CNPRJTXDIHRZPF
|
6.2 | Ki | 4 | — | |
UUDTVMMARAFNKG
|
6.2 | Ki | 4 | — | |
PYKDJHBKQBUYDN
|
6.2 | IC50 | 2 | — | |
BBMXXNQSDJPWKT
|
6.2 | IC50 | 4 | — | |
GIEQMQWMJSYCKB
|
6.2 | Ki | 5 | — | |
BFJIOGLKGISOKV
|
6.2 | Ki | 8 | — | |
QTTXNAZRANVJPE
|
6.2 | IC50 | 2 | — | |
WQJPTWWOCNRCBI
|
6.2 | IC50 | 2 | — | |
GWHSSPUFNDIEEQ
|
6.1 | Ki | 4 | — | |
VPRBKPRUOSPYMW
|
6.1 | IC50 | 2 | — | |
WTCSNHGGDSKNJP
|
6.1 | IC50 | 2 | — | |
MMIHYNVQXYWTFM
|
6.1 | Ki | 4 | — | |
KLSPLBHGNYWPLX
|
6.1 | IC50 | 3 | — | |
UWVBDELWTIGPFO
|
6.1 | Ki | 4 | — | |
BLDFRIYOIZRRJI
|
6.1 | Ki | 4 | — | |
MMIHYNVQXYWTFM
|
6.1 | Ki | 4 | — | |
UGWWPGUNBPZMDD
|
6.0 | IC50 | 5 | — | |
RUVHVYMIMBVNKN
|
6.0 | Ki | 5 | — | |
LXZKIXQSLYEDMA
|
6.0 | IC50 | 2 | — | |
LXZKIXQSLYEDMA
|
6.0 | IC50 | 2 | — |