Target Details
| UniProt AC | P09238 |
|---|---|
| Gene Symbol | MMP10 |
| Protein Name | Stromelysin-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 133
- Clinical molecules 5
- Avg pChEMBL 6.99
Active Molecules (133)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IWQSGINKBSWILJ
|
9.5 | IC50 | 10 | — | |
HXZPYZWICHZKRL
|
9.5 | IC50 | 10 | — | |
ROSNVSQTEGHUKU
|
9.3 | IC50 | 12 | Yes | |
VBMQORMYXJZHKU
|
8.8 | Ki | 2 | — | |
CUKATAAPVFYVIL
|
8.6 | IC50 | 9 | — | |
JGWTVBVOISUVJD
|
8.6 | IC50 | 9 | — | |
JVKDGTTXLCSABF
|
8.5 | IC50 | 2 | — | |
PJTIDEQBVYCKIC
|
8.4 | IC50 | 2 | — | |
FMEMUXYNXWETSE
|
8.2 | IC50 | 6 | — | |
BJBBGWSFUXQTAD
|
8.2 | IC50 | 2 | — | |
JHSGRRNCQDDQBC
|
8.1 | IC50 | 9 | — | |
OUZMHHWAGJCAFA
|
8.1 | Ki | 8 | — | |
PTUCPHGSAFOJAU
|
8.1 | Ki | 9 | — | |
DYBVZAZWVGRLPI
|
8.1 | IC50 | 2 | — | |
GHWPTWVNZOSEBR
|
7.9 | IC50 | 2 | — | |
ZUZGJCNWNOCKEB
|
7.9 | IC50 | 2 | — | |
CQORHEXIKLKTGU
|
7.9 | IC50 | 2 | — | |
ZGBAPSHWPBXEKN
|
7.9 | IC50 | 10 | — | |
FIQXBPSAOMLPLJ
|
7.8 | IC50 | 2 | — | |
VUEMJXMTPAGVNJ
|
7.8 | IC50 | 2 | — | |
ZQKGUWOTJVDTGX
|
7.8 | IC50 | 2 | — | |
ZUZGJCNWNOCKEB
|
7.8 | IC50 | 2 | — | |
AYPBWVMVAOAQCE
|
7.7 | IC50 | 2 | — | |
ZUZGJCNWNOCKEB
|
7.7 | IC50 | 2 | — | |
ISAKGERLXJBHSA
|
7.6 | IC50 | 2 | — | |
WJUVUTHXZGHZOG
|
7.6 | IC50 | 2 | — | |
UFKJDXKTPYNZRZ
|
7.5 | IC50 | 4 | — | |
XHWPSFKZEOYPJH
|
7.5 | IC50 | 2 | — | |
MVYFKOXRGAPNAN
|
7.5 | IC50 | 2 | — | |
HGMNWCDIIMBGAR
|
7.5 | IC50 | 4 | — | |
QCVLVTVGVJUODZ
|
7.5 | Ki | 6 | — | |
XHPUXKQBUUHEIP
|
7.5 | Ki | 6 | — | |
ZWXRGJMHGHMUMB
|
7.4 | Ki | 4 | — | |
XGAABSVAAOEGKA
|
7.4 | IC50 | 2 | — | |
KOVQMCGGWATESY
|
7.4 | Ki | 6 | — | |
OIZMOMFOLNBXHF
|
7.3 | IC50 | 9 | — | |
KOVQMCGGWATESY
|
7.3 | Ki | 7 | — | |
KMXAXPCBRVZOGA
|
7.3 | IC50 | 7 | — | |
LFUNCOOVDREPBK
|
7.3 | Ki | 6 | — | |
KIMPOJXDFKFBTL
|
7.3 | IC50 | 2 | — | |
KNOYHJOPRUTPSQ
|
7.3 | Ki | 7 | — | |
RCSJFBBGCSVIIU
|
7.3 | IC50 | 2 | — | |
MLUCCAMJMIYYED
|
7.3 | IC50 | 3 | — | |
LTJSRJHCFOHUDW
|
7.2 | IC50 | 2 | — | |
YXPTXTBBPCLWPQ
|
7.2 | IC50 | 4 | — | |
NKVXPWMSTSLIPX
|
7.2 | IC50 | 2 | — | |
OCSMOTCMPXTDND
|
7.2 | IC50 | 14 | Yes | |
ZQUJAHCTHDEZMJ
|
7.2 | Ki | 6 | — | |
MXFJZXDWWXHXMV
|
7.1 | Ki | 7 | — | |
NIAIEBGBRXKPAO
|
7.1 | Ki | 7 | — |