Target Details
| UniProt AC | P09237 |
|---|---|
| Gene Symbol | MMP7 |
| Protein Name | Matrilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 241
- Clinical molecules 184
- Avg pChEMBL 7.11
KEGG Pathways (2)
Active Molecules (241)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CRPDTHYTIJXWLZ
|
6.2 | IC50 | 7 | Yes | |
MTGNBEKVSCTMSE
|
6.2 | IC50 | 5 | Yes | |
KCBXQUWPZNVZIG
|
6.1 | Ki | 2 | — | |
NWAZOLPVSMLDTN
|
6.1 | IC50 | 5 | Yes | |
XDYZXHJJAIXYOR
|
6.1 | IC50 | 8 | Yes | |
BUOKQWSUTKFXOW
|
6.1 | IC50 | 6 | Yes | |
GPLRECXXBJTJRJ
|
6.1 | IC50 | 6 | Yes | |
RCXJWFMVFQBLSC
|
6.1 | IC50 | 8 | Yes | |
IAENNQHKVZEBQT
|
6.1 | IC50 | 7 | Yes | |
ITNSNSYBFZWVPE
|
6.1 | IC50 | 5 | Yes | |
JRZMGNCXDSZZAF
|
6.1 | Ki | 3 | — | |
YGXMCNARAMUPPX
|
6.1 | IC50 | 7 | Yes | |
DYVJPNSKJGHBKT
|
6.1 | IC50 | 6 | Yes | |
IWJCPVCPLCTWHT
|
6.1 | IC50 | 5 | Yes | |
OIZMOMFOLNBXHF
|
6.1 | IC50 | 9 | — | |
PCRITYAGTCCZEK
|
6.1 | Ki | 7 | Yes | |
RWKJBOMUESGCBO
|
6.1 | Ki | 4 | Yes | |
AKWKBACKRMYPRV
|
6.1 | Ki | 6 | Yes | |
BTZXQMHZPVTFBL
|
6.1 | IC50 | 7 | Yes | |
IIDUBAKXXSWORH
|
6.1 | IC50 | 5 | Yes | |
NACPMNMCCDZXLH
|
6.1 | IC50 | 6 | Yes | |
QLMFPICUYDVBBS
|
6.1 | IC50 | 4 | — | |
HHHAELOQIYTSIY
|
6.1 | IC50 | 6 | Yes | |
HXAROWWJPCDNRW
|
6.0 | IC50 | 6 | Yes | |
KGUVBHLPMGERAT
|
6.0 | IC50 | 8 | Yes | |
CPBPQYOAJUZJNL
|
6.0 | IC50 | 7 | Yes | |
KKVTZTBYJGHGCO
|
6.0 | IC50 | 8 | Yes | |
QKXUIPRJJWLPIY
|
6.0 | IC50 | 7 | Yes | |
VAQNHYAKIUNIKM
|
6.0 | IC50 | 8 | Yes | |
YVUNEHSVUBACDW
|
6.0 | IC50 | 6 | Yes | |
IMKDKHQDFFLOKK
|
6.0 | IC50 | 13 | Yes | |
KXZZWRQJKQVMKR
|
6.0 | IC50 | 7 | Yes | |
VMOSDDURWLNMNG
|
6.0 | IC50 | 8 | Yes | |
LIQFLIXIOKMDTJ
|
6.0 | Ki | 7 | Yes | |
YNIHTMMJQXUNPE
|
6.0 | Ki | 7 | Yes | |
CUKATAAPVFYVIL
|
6.0 | IC50 | 9 | — | |
DABGHULKCXXLEE
|
6.0 | IC50 | 4 | — | |
GQLPTZZPKXZFQR
|
6.0 | Ki | 5 | Yes | |
OKHKINWJYOOKOF
|
6.0 | IC50 | 3 | — | |
SXFDETGXHVKYJE
|
6.0 | IC50 | 6 | Yes | |
YBPDYJXZXAPGSU
|
6.0 | IC50 | 6 | Yes |