Target Details
| UniProt AC | P09237 |
|---|---|
| Gene Symbol | MMP7 |
| Protein Name | Matrilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 241
- Clinical molecules 184
- Avg pChEMBL 7.11
KEGG Pathways (2)
Active Molecules (241)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WFVYENBQHIIIQE
|
6.5 | IC50 | 7 | Yes | |
TYZVGHNHMXVHTN
|
6.5 | Ki | 5 | — | |
SEQZHNNPDSVBRC
|
6.5 | IC50 | 6 | Yes | |
AWPBSKGASHYAHG
|
6.5 | IC50 | 5 | Yes | |
IIKWXGAHGMGLSQ
|
6.5 | IC50 | 3 | — | |
VDUBALDTEGAJSW
|
6.5 | Ki | 7 | Yes | |
YTCCTPYUECNUFO
|
6.5 | IC50 | 7 | Yes | |
CMBPIMDJJHAVBX
|
6.4 | IC50 | 6 | Yes | |
HTNLSTWGHBHDPS
|
6.4 | IC50 | 8 | Yes | |
NFDNOGJHVSTSMJ
|
6.4 | Ki | 7 | Yes | |
NVNGYUBMJMOHQL
|
6.4 | IC50 | 6 | Yes | |
DEZZFUOGAFLCST
|
6.4 | IC50 | 6 | Yes | |
DOIKBNWTWCOTKR
|
6.4 | IC50 | 7 | Yes | |
GWZMHEYDUOAMNJ
|
6.4 | IC50 | 6 | Yes | |
BJOZETKUSDMMAN
|
6.4 | IC50 | 6 | Yes | |
QGTWMCXPSZIGIN
|
6.3 | IC50 | 6 | Yes | |
RVKPGECPCLBLDB
|
6.3 | IC50 | 10 | Yes | |
BCWUIVYEXBBRHO
|
6.3 | IC50 | 6 | Yes | |
BZVYQWLRCHLAGK
|
6.3 | IC50 | 10 | Yes | |
USIMDPVZFWUXPH
|
6.3 | IC50 | 6 | Yes | |
QVNZBDLTUKCPGJ
|
6.3 | IC50 | 10 | — | |
QYFKTMNLZHLRIH
|
6.3 | IC50 | 7 | Yes | |
RYRSPABEKSPRKC
|
6.3 | IC50 | 7 | Yes | |
UBBBKPVDKLDZNE
|
6.3 | IC50 | 7 | Yes | |
AMOCYMNNMVOHOG
|
6.3 | IC50 | 6 | Yes | |
GWXMWHCYBJJJND
|
6.3 | IC50 | 6 | Yes | |
JDOCJRYXQAWUOO
|
6.3 | IC50 | 7 | Yes | |
MXFJZXDWWXHXMV
|
6.3 | Ki | 7 | — | |
ODFXJYBYTABKHA
|
6.3 | IC50 | 7 | Yes | |
ZFYWVXBCKVCYOL
|
6.3 | IC50 | 7 | Yes | |
XGJAXXYDMLECBQ
|
6.3 | IC50 | 7 | Yes | |
TZQQXIZDSZWWPC
|
6.3 | IC50 | 6 | Yes | |
KEWGKOQZKWDXBX
|
6.3 | IC50 | 7 | Yes | |
PYNQNWZHEDOQHX
|
6.3 | IC50 | 6 | Yes | |
NTWPNMLRTBRVIB
|
6.2 | IC50 | 5 | Yes | |
RFNUTMXSNZMOSL
|
6.2 | Ki | 7 | Yes | |
ZGBAPSHWPBXEKN
|
6.2 | IC50 | 10 | — | |
ZUAZPXLMAVHRDA
|
6.2 | Ki | 3 | — | |
HAIGFFSNUYJTQK
|
6.2 | IC50 | 6 | Yes | |
IQUZJJXEDANMJD
|
6.2 | Ki | 4 | — | |
KJBQTISDZZFFDE
|
6.2 | IC50 | 5 | Yes | |
OECFBMNWNGPPFC
|
6.2 | IC50 | 6 | Yes | |
BPNDGQNQHSBNOE
|
6.2 | IC50 | 7 | Yes | |
BYQIIKCYPGKHOY
|
6.2 | Ki | 5 | Yes | |
PTUCPHGSAFOJAU
|
6.2 | Ki | 9 | — | |
PTUCPHGSAFOJAU
|
6.2 | Ki | 9 | Yes | |
PTUCPHGSAFOJAU
|
6.2 | Ki | 7 | — | |
INSQINPAEQOIQL
|
6.2 | IC50 | 7 | Yes | |
WICQDDCNCVTFDX
|
6.2 | Ki | 16 | Yes | |
VXVNMUQIRGITQV
|
6.2 | IC50 | 5 | Yes |