Target Details
| UniProt AC | P09237 |
|---|---|
| Gene Symbol | MMP7 |
| Protein Name | Matrilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 241
- Clinical molecules 184
- Avg pChEMBL 7.11
KEGG Pathways (2)
Active Molecules (241)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
USIBDKCJHKIPNX
|
7.2 | IC50 | 6 | Yes | |
YKPYIPVDTNNYCN
|
7.2 | IC50 | 11 | Yes | |
IZXYSBTXZXSNBA
|
7.2 | IC50 | 6 | Yes | |
JHSGRRNCQDDQBC
|
7.2 | IC50 | 9 | — | |
NDOOKPHRXLOQEK
|
7.2 | IC50 | 4 | Yes | |
HJNKYGBTSGQBDU
|
7.1 | Ki | 10 | — | |
UDNLRUDZHBXCON
|
7.1 | Ki | 7 | Yes | |
RMKNDVDQYWXAON
|
7.1 | IC50 | 7 | Yes | |
RYMINZKMUZXTLF
|
7.1 | IC50 | 6 | Yes | |
GETQXLAMYOMSJS
|
7.1 | IC50 | 8 | Yes | |
OCZKLINSAMKTBK
|
7.0 | IC50 | 7 | Yes | |
WSFQQGCWUCOARG
|
7.0 | Ki | 6 | — | |
GAQJSKIBXSLAJK
|
7.0 | IC50 | 6 | Yes | |
BSIZUMJRKYHEBR
|
7.0 | IC50 | 15 | Yes | |
DUONGMKIDQRGNH
|
7.0 | IC50 | 6 | — | |
KMLOBHZAEFITDB
|
7.0 | IC50 | 4 | — | |
NIPJJOWPCLBDGS
|
7.0 | IC50 | 8 | Yes | |
RTSLKKUJJKXEJT
|
7.0 | IC50 | 5 | Yes | |
YKHOQKKUOWOUDP
|
6.9 | Ki | 2 | — | |
RIOJMNDNYHZZFM
|
6.9 | Ki | 7 | Yes | |
XWGUPBCCRWJAMM
|
6.9 | IC50 | 6 | Yes | |
VHCRBJFCQRNNFG
|
6.8 | IC50 | 8 | Yes | |
CJTUBZULFXKTAT
|
6.8 | IC50 | 10 | Yes | |
TUSYEXLVYIINDP
|
6.8 | IC50 | 6 | Yes | |
DQLDJYJWPVFOFC
|
6.8 | Ki | 7 | Yes | |
BQDVTMRZPWSYOT
|
6.7 | IC50 | 7 | — | |
CIQJGNDHWOIZCK
|
6.7 | IC50 | 6 | Yes | |
NQPIHEUUYRAYII
|
6.7 | IC50 | 8 | Yes | |
ZHLANTZRDCBWFM
|
6.7 | IC50 | 6 | Yes | |
JYUUAPXGAQJXBY
|
6.7 | IC50 | 3 | — | |
KUDBVBLUURDAMX
|
6.7 | IC50 | 5 | Yes | |
JGRIYRSQHHLUHI
|
6.7 | IC50 | 7 | Yes | |
WXMUXNHNFVCNMU
|
6.7 | IC50 | 5 | — | |
LZUHYMGQNXWOHQ
|
6.7 | IC50 | 6 | — | |
ROSNVSQTEGHUKU
|
6.7 | IC50 | 12 | Yes | |
ZGTPJERIIBYCFG
|
6.7 | Ki | 5 | Yes | |
GCGWPKSFLVGEQR
|
6.7 | IC50 | 4 | Yes | |
BSTYDWORGHMRLI
|
6.6 | Ki | 5 | — | |
DNGGPLKVDUPXFN
|
6.6 | IC50 | 5 | — | |
DNGGPLKVDUPXFN
|
6.6 | IC50 | 7 | Yes | |
UKLIIGXGTPSYBF
|
6.6 | IC50 | 8 | Yes | |
YPKIDRAXEHHNGA
|
6.6 | Ki | 2 | — | |
YDMIPBHQKFOFQW
|
6.6 | Ki | 7 | Yes | |
WXUQPWYPRTYWIR
|
6.6 | IC50 | 6 | Yes | |
LUHJAOVICRNTRC
|
6.5 | IC50 | 7 | Yes | |
FIAWLFURFKPROF
|
6.5 | IC50 | 7 | Yes | |
BKIYUSXBJJEODV
|
6.5 | IC50 | 7 | Yes | |
JMKHBHJIGFWJPF
|
6.5 | IC50 | 5 | — | |
NWVCPUQBLORAAX
|
6.5 | IC50 | 3 | — | |
YIYXDKFJIKECAM
|
6.5 | IC50 | 5 | Yes |