Target Details
| UniProt AC | P09237 |
|---|---|
| Gene Symbol | MMP7 |
| Protein Name | Matrilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 241
- Clinical molecules 184
- Avg pChEMBL 7.11
KEGG Pathways (2)
Active Molecules (241)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVBJVUYVRZYYHC
|
8.0 | IC50 | 5 | Yes | |
DDRBOOUOUSFWET
|
8.0 | IC50 | 4 | — | |
GKHRDWHFKKUYAX
|
8.0 | IC50 | 8 | Yes | |
MHQJDNZHPIZRRV
|
8.0 | IC50 | 4 | — | |
OCSMOTCMPXTDND
|
8.0 | IC50 | 14 | Yes | |
RYDPXGZLAKQPJB
|
8.0 | Ki | 6 | — | |
QDPILJAKSNERSV
|
7.9 | Ki | 6 | — | |
LPRBYIANGHPFSM
|
7.9 | IC50 | 4 | Yes | |
CKCBYWFMRXPHJM
|
7.8 | Ki | 4 | — | |
PZPOCZWOYXDPDG
|
7.8 | IC50 | 5 | Yes | |
XSWDEIOVOAQSMZ
|
7.8 | IC50 | 7 | Yes | |
IXHBDLPZTUSLFD
|
7.8 | Ki | 5 | — | |
WMYJDFANEQLDGP
|
7.8 | IC50 | 6 | — | |
BODLESUVCQEUII
|
7.7 | Ki | 7 | Yes | |
IZYWROOEWSDARX
|
7.7 | Ki | 6 | Yes | |
KJVHFBOUABDIQV
|
7.7 | IC50 | 5 | Yes | |
TVNINFNNQVBJHI
|
7.7 | IC50 | 8 | Yes | |
GFUITADOEPNRML
|
7.7 | IC50 | 11 | Yes | |
OCSMOTCMPXTDND
|
7.7 | IC50 | 8 | Yes | |
SSNRGEULLFASJG
|
7.7 | IC50 | 4 | Yes | |
YUWSFQQPCKKPJG
|
7.7 | IC50 | 9 | Yes | |
GTXSRFUZSLTDFX
|
7.6 | IC50 | 8 | Yes | |
ULILDPSFFUSXJH
|
7.6 | IC50 | 9 | Yes | |
ULILDPSFFUSXJH
|
7.6 | IC50 | 7 | — | |
HYBHKZKKEGAPOP
|
7.6 | IC50 | 6 | — | |
ANFAAJVPGXQKBB
|
7.6 | IC50 | 6 | Yes | |
NUVSGXIVCJBRBF
|
7.6 | Ki | 3 | — | |
CVZIHNYAZLXRRS
|
7.6 | IC50 | 10 | Yes | |
NOXYNXIAEWTFQX
|
7.6 | IC50 | 7 | Yes | |
SGQBRJNZCHCINW
|
7.5 | IC50 | 6 | Yes | |
AKNDZTHCJLFZCF
|
7.5 | IC50 | 9 | Yes | |
CYYCSKFJEOSZTF
|
7.5 | IC50 | 9 | Yes | |
HXZPYZWICHZKRL
|
7.5 | IC50 | 10 | — | |
MCSWSPNUKWMZHM
|
7.5 | IC50 | 7 | Yes | |
QYZPDCGWIJYZMN
|
7.5 | IC50 | 8 | Yes | |
NITYDPDXAAFEIT
|
7.5 | IC50 | 20 | Yes | |
YZOKWMYHTLQIDP
|
7.5 | IC50 | 5 | Yes | |
XXOLBMKULOJKQR
|
7.4 | IC50 | 7 | Yes | |
PYXPFZLYNSTHAH
|
7.4 | Ki | 4 | — | |
XJMLKUIRAXOATH
|
7.4 | IC50 | 7 | Yes | |
YLQBSSFZOXXRNR
|
7.4 | IC50 | 6 | Yes | |
QESYNYYOSNECPA
|
7.4 | IC50 | 6 | Yes | |
CQRAUIRVDKNRIO
|
7.4 | IC50 | 9 | Yes | |
GKHRDWHFKKUYAX
|
7.4 | IC50 | 9 | — | |
DOECLBQWTWHNID
|
7.3 | IC50 | 4 | Yes | |
KJNZDUKNEQXTSO
|
7.3 | Ki | 6 | — | |
TUXGRLPRNXNACO
|
7.3 | IC50 | 5 | Yes | |
CYBDDZKSRZPTQR
|
7.3 | IC50 | 6 | Yes | |
KMLOBHZAEFITDB
|
7.3 | IC50 | 4 | — | |
WIUDGBCTJVXBCM
|
7.3 | IC50 | 7 | — |