Target Details
| UniProt AC | P09237 |
|---|---|
| Gene Symbol | MMP7 |
| Protein Name | Matrilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 241
- Clinical molecules 184
- Avg pChEMBL 7.11
KEGG Pathways (2)
Active Molecules (241)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YQYRZEZDMHAWCC
|
9.8 | IC50 | 2 | — | |
CEEASCNCHQSPKF
|
9.6 | IC50 | 5 | Yes | |
QVHQLFLTQMCYLJ
|
9.5 | IC50 | 6 | Yes | |
AAPPTEGQHHRRCP
|
9.1 | IC50 | 6 | Yes | |
HFAGTNGCAZYYLZ
|
9.1 | Ki | 13 | Yes | |
JCVSSJUXUIJGBT
|
9.0 | IC50 | 5 | Yes | |
YIJAXOAFVMWOOR
|
9.0 | IC50 | 5 | Yes | |
IOTJDDOXTYOJJN
|
9.0 | IC50 | 6 | Yes | |
JMYNELQJPYBCPZ
|
8.9 | IC50 | 6 | Yes | |
DONMTDNLNMLOIC
|
8.8 | Ki | 13 | Yes | |
ZAXDLNVDZOYNCA
|
8.8 | IC50 | 6 | Yes | |
BJOZETKUSDMMAN
|
8.8 | IC50 | 6 | Yes | |
XEONYLBJVDXPRB
|
8.8 | IC50 | 6 | Yes | |
OCQHJTWHXNLSJE
|
8.7 | IC50 | 5 | Yes | |
PJKWYBIJVPNFJI
|
8.7 | IC50 | 6 | Yes | |
VYGKNAIULXUTGK
|
8.7 | IC50 | 6 | Yes | |
QPPXLNJKZJGLRN
|
8.6 | IC50 | 6 | Yes | |
ITXQTOBRXFVFDQ
|
8.6 | IC50 | 2 | — | |
YKYLOHCKSMYHPL
|
8.6 | IC50 | 6 | Yes | |
GCBPAPVOMPJQHK
|
8.5 | Ki | 9 | Yes | |
USEJKZYMWYHGSP
|
8.5 | IC50 | 7 | Yes | |
FVGUURIXHJHLQF
|
8.5 | IC50 | 4 | Yes | |
QQWABDFFKSDQLH
|
8.5 | IC50 | 6 | Yes | |
JQYSJWITJMOASO
|
8.5 | IC50 | 6 | Yes | |
AALOSJKQIIRSAO
|
8.4 | IC50 | 6 | Yes | |
KDIPAKUGVJEBFC
|
8.4 | IC50 | 2 | — | |
XFILPEOLDIKJHX
|
8.4 | IC50 | 12 | Yes | |
LBZOGBFXCHOCBC
|
8.4 | IC50 | 6 | Yes | |
UERCGTJUVRFNRO
|
8.4 | Ki | 6 | Yes | |
BZTWELLPCHJZLB
|
8.4 | IC50 | 6 | Yes | |
FXEYKJYOHRTUNG
|
8.4 | IC50 | 6 | Yes | |
HEPINVNDBLHRTM
|
8.4 | IC50 | 6 | Yes | |
DZVQTAQHEPKNSI
|
8.4 | IC50 | 6 | Yes | |
OONXADPQRATYFL
|
8.3 | Ki | 5 | Yes | |
WORSVFBVUCBRIP
|
8.3 | IC50 | 5 | — | |
IKIPPVJMYSOQOD
|
8.2 | IC50 | 6 | Yes | |
VCJOCQOXJUMEBE
|
8.2 | IC50 | 6 | Yes | |
RGQWTGAVFAYQEF
|
8.2 | IC50 | 6 | Yes | |
FPSMXPGSVWPWCG
|
8.2 | IC50 | 8 | — | |
SIICAQVADMFEDB
|
8.2 | Ki | 8 | Yes | |
IWQSGINKBSWILJ
|
8.1 | IC50 | 10 | — | |
WVSIAOYHEIZRMM
|
8.1 | IC50 | 2 | — | |
DXDRHHKMWQZJHT
|
8.1 | IC50 | 9 | — | |
LXWSFODDORIHFJ
|
8.1 | IC50 | 6 | Yes | |
MOPRTFSMCQNUCT
|
8.1 | IC50 | 9 | Yes | |
NMPGSGFXAAVWRZ
|
8.1 | IC50 | 2 | — | |
YLXVWRCBKXEQFD
|
8.1 | IC50 | 6 | Yes | |
HOGIHVAAHRAULF
|
8.0 | IC50 | 5 | Yes | |
QTHGVXWBMQNWSU
|
8.0 | IC50 | 2 | — | |
QVXRAVFETVTALN
|
8.0 | IC50 | 5 | Yes |