Target Details
| UniProt AC | P09038 |
|---|---|
| Gene Symbol | FGF2 |
| Protein Name | Fibroblast growth factor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00167 (FGF) |
Summary
- Multi-target molecules 69
- Clinical molecules 0
- Avg pChEMBL 6.76
KEGG Pathways (15)
- Breast cancer
- Calcium signaling pathway
- Chemical carcinogenesis - receptor activation
- EGFR tyrosine kinase inhibitor resistance
- Gastric cancer
- Kaposi sarcoma-associated herpesvirus infection
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
Active Molecules (69)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BQWLMOMUMNGHQA
|
6.3 | Kd | 2 | — | |
GJRDMRRBRLWIMA
|
6.3 | IC50 | 4 | — | |
LCULSEGLGJAWDH
|
6.3 | Kd | 3 | — | |
MIKHBYRVCGYIJG
|
6.3 | Kd | 3 | — | |
MTFFLFAICAKCHG
|
6.3 | Kd | 3 | — | |
GQXXCBAPTBXUNH
|
6.3 | Kd | 3 | — | |
FDSOODAZYPJSDK
|
6.3 | IC50 | 4 | — | |
CAQCMXFJWJJJLH
|
6.3 | IC50 | 4 | — | |
OBNDKQCXTGZBFN
|
6.3 | Kd | 3 | — | |
RBWDOUOLUKRISD
|
6.3 | Kd | 4 | — | |
VENGQIUBROEMGG
|
6.3 | Kd | 3 | — | |
UXXWCLFQFHSDIF
|
6.2 | IC50 | 4 | — | |
NRKBLKNBNMFJGW
|
6.2 | IC50 | 4 | — | |
XTCMHHNUPIPYQB
|
6.2 | IC50 | 4 | — | |
ZZZNJDODCKXBLN
|
6.2 | IC50 | 4 | — | |
KTWJKWUVFXXMTI
|
6.2 | IC50 | 4 | — | |
SUXXKYXDLFQQTP
|
6.2 | IC50 | 4 | — | |
ODJIBJUXPSKWRB
|
6.2 | Kd | 3 | — | |
IPWXMKVZKOEZQH
|
6.2 | Kd | 3 | — |