Target Details
| UniProt AC | P08922 |
|---|---|
| Gene Symbol | ROS1 |
| Protein Name | Proto-oncogene tyrosine-protein kinase ROS |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 263
- Clinical molecules 18
- Avg pChEMBL 7.6
Associated Diseases (1)
Active Molecules (263)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HXHAJRMTJXHJJZ
|
6.0 | Ki | 52 | Yes | |
IIIJQZOSLLAVTL
|
6.0 | Ki | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MMMPFWNSQKXKDX
|
6.0 | Ki | 14 | — | |
NHFDRBXTEDBWCZ
|
6.0 | Ki | 41 | — | |
NRGYZNJPCGRCLV
|
6.0 | Ki | 52 | — | |
PRRYQINUAIQTFJ
|
6.0 | Ki | 11 | — | |
UZWDCWONPYILKI
|
6.0 | IC50 | 47 | — | |
VXYDJXMHISGSDA
|
6.0 | Ki | 59 | — | |
WFTZMAAMCVPJJT
|
6.0 | Ki | 26 | — | |
ZEWQUBUPAILYHI
|
6.0 | IC50 | 21 | — |