Target Details
| UniProt AC | P08922 |
|---|---|
| Gene Symbol | ROS1 |
| Protein Name | Proto-oncogene tyrosine-protein kinase ROS |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 263
- Clinical molecules 18
- Avg pChEMBL 7.6
Associated Diseases (1)
Active Molecules (263)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WVXNSAVVKYZVOE
|
6.5 | IC50 | 92 | — | |
IJVDETPCUCZHTR
|
6.4 | Ki | 12 | — | |
JXNMCDLXYWQTIW
|
6.4 | Ki | 13 | — | |
NRSGWEVTVGZDFC
|
6.4 | Ki | 50 | — | |
PBZAJAZDOFEDDH
|
6.4 | IC50 | 2 | — | |
PTVPBWWDGZSEAF
|
6.4 | Ki | 63 | — | |
QNUKRWAIZMBVCU
|
6.4 | Ki | 46 | — | |
UMTWTCVTRDYHQQ
|
6.4 | Ki | 56 | — | |
VEPKQEUBKLEPRA
|
6.4 | Ki | 11 | — | |
QLAIBBCRJCMGRY
|
6.4 | Kd | 2 | — | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 91 | Yes | |
CLRFYTGANQZOBS
|
6.3 | Ki | 41 | — | |
IFQICUARAXVEIQ
|
6.3 | Ki | 18 | — | |
KDKUVYLMPJIGKA
|
6.3 | Ki | 91 | Yes | |
LRINYHMQZRENCY
|
6.3 | Ki | 29 | — | |
JQWJRFOFKDLCQB
|
6.3 | IC50 | 2 | — | |
ZQTNTFAUQJEQHU
|
6.2 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
RKERQEKFTWWCEY
|
6.2 | IC50 | 4 | — | |
GCIKSSRWRFVXBI
|
6.2 | Kd | 109 | Yes | |
CHTMRWQLNNRRFJ
|
6.2 | Ki | 70 | — | |
DBKQWGCVGCVPIP
|
6.2 | Ki | 21 | — | |
FQBWBTKXLRVHDG
|
6.2 | Ki | 3 | — | |
GLMWKEAUVZDGKE
|
6.2 | Ki | 23 | — | |
NJPWCTYVEJIQBM
|
6.2 | Ki | 72 | — | |
OADRBDVURCEKRP
|
6.2 | Ki | 44 | — | |
PUPCRRRSBUYJAD
|
6.2 | Ki | 44 | Yes | |
VBUWAJWPXASNGM
|
6.2 | Ki | 9 | — | |
XBDWKVLCDCUNHH
|
6.2 | Ki | 18 | — | |
XHORJSJFHVABEA
|
6.2 | Ki | 49 | — | |
XYZNKCSDQRKAFR
|
6.2 | Ki | 53 | — | |
YKYRQCWLYUTVIE
|
6.2 | Ki | 16 | — | |
VDXGLZJPQRGNLY
|
6.1 | IC50 | 10 | — | |
BZFGDXJGWSIYQP
|
6.1 | Ki | 9 | — | |
CQXFMKMVOOUGSS
|
6.1 | Ki | 6 | — | |
HHFBDROWDBDFBR
|
6.1 | Ki | 40 | Yes | |
IJRBJCMLWLFMIN
|
6.1 | Ki | 17 | — | |
IZAVTOABECKIDH
|
6.1 | Ki | 20 | — | |
OMKZJNFKGWJFNX
|
6.1 | Ki | 8 | — | |
OUJZYQBEFNDJQN
|
6.1 | Ki | 71 | — | |
PCQMERRARZKTPW
|
6.1 | Ki | 68 | — | |
SVUIYNKSDCANAY
|
6.1 | Ki | 16 | — | |
YUOWJICKAJQZLS
|
6.1 | Ki | 35 | — | |
YWTBGJGMTBHQTM
|
6.1 | Ki | 65 | — | |
CUIHSIWYWATEQL
|
6.0 | Kd | 61 | Yes | |
BSFNGHCTZDCQBF
|
6.0 | Ki | 93 | — | |
CXBBWVXSZINRCS
|
6.0 | Ki | 41 | — | |
FDVSOQRNTAPCHB
|
6.0 | Ki | 40 | — | |
GDLIGKIOYRNHDA
|
6.0 | IC50 | 24 | Yes |