Target Details
| UniProt AC | P08922 |
|---|---|
| Gene Symbol | ROS1 |
| Protein Name | Proto-oncogene tyrosine-protein kinase ROS |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 263
- Clinical molecules 18
- Avg pChEMBL 7.6
Associated Diseases (1)
Active Molecules (263)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LYNBNVBMAGDJRW
|
7.2 | Ki | 81 | — | |
MVJMMLFMPWITEJ
|
7.2 | Ki | 110 | — | |
VQPBIJGXSXEOCU
|
7.2 | Ki | 24 | — | |
ZBXKQGMXXMNDQF
|
7.2 | IC50 | 2 | — | |
GLDSKRNGVVYJAB
|
7.1 | Kd | 16 | — | |
SGZZQKMOFHIDKW
|
7.1 | Kd | 13 | — | |
DFMCXVONDDGQIY
|
7.1 | Ki | 66 | — | |
GCBJDOWIQHMCMR
|
7.1 | Ki | 84 | — | |
GDYZFFBMSBDTAA
|
7.1 | Ki | 60 | — | |
YMIJUBCSOKSFRU
|
7.1 | Ki | 87 | — | |
ZKHDDJKHTPLPOQ
|
7.1 | Ki | 62 | — | |
OMVJEQVEBCZADZ
|
7.1 | IC50 | 3 | — | |
VPYPBQZXCLHXPF
|
7.1 | IC50 | 3 | — | |
CWBWMDSAVFJNAD
|
7.0 | Ki | 7 | — | |
VKBFHTIUXUCYRQ
|
7.0 | Ki | 66 | — | |
VFWZEMIPXRZJDU
|
7.0 | IC50 | 2 | — | |
KRHJQHMWPVTYCU
|
7.0 | IC50 | 6 | — | |
YLCFOHVAOBLAIK
|
7.0 | IC50 | 14 | — | |
FPQNRXITKTZFMF
|
6.9 | Kd | 13 | — | |
DSSRVQAIWBZWON
|
6.9 | Ki | 9 | — | |
FQEODTMNWMDUMD
|
6.8 | Ki | 25 | — | |
FUMCKNCUEAQHCV
|
6.8 | Ki | 103 | — | |
GXJSLIOOPZRPEV
|
6.8 | Ki | 34 | — | |
NLUPJKQOKWBWFC
|
6.8 | Ki | 69 | — | |
RTDSHUGNRVXRHN
|
6.8 | Ki | 51 | — | |
ZLHFILGSQDJULK
|
6.8 | Ki | 37 | Yes | |
ZLVOTRRGLSDLPF
|
6.8 | Ki | 36 | — | |
UMBIRSZUCJNBHB
|
6.8 | IC50 | 18 | — | |
BLQYVHBZHAISJM
|
6.7 | Ki | 54 | — | |
IOBVCHJTLVPPBR
|
6.7 | Ki | 39 | — | |
LRZYYIZFBXFSJB
|
6.7 | Ki | 69 | — | |
MASJMHFQMYAPJR
|
6.7 | Ki | 41 | — | |
UBPYILGKFZZVDX
|
6.7 | IC50 | 130 | Yes | |
XNRABRXYGRUDAX
|
6.7 | IC50 | 3 | — | |
ZXLFIHLBHMLHFJ
|
6.7 | Ki | 31 | — | |
QSGGLLCPVRJDDE
|
6.7 | IC50 | 4 | — | |
NXSJMRCTGYTSTK
|
6.6 | Kd | 200 | — | |
BIIVYFLTOXDAOV
|
6.6 | Ki | 31 | — | |
NPJROAJIXPVMTE
|
6.6 | Ki | 8 | — | |
QONPPIZSNSSCSK
|
6.6 | Ki | 45 | Yes | |
VNGYQBMDQMDALH
|
6.6 | Ki | 25 | — | |
GCDSDVNITVBCDW
|
6.6 | IC50 | 17 | — | |
UEBRHNWRYCBULZ
|
6.6 | Ki | 2 | — | |
OXQTXNVWTNDAQF
|
6.5 | IC50 | 5 | — | |
AAYZTFLAQXDFOL
|
6.5 | Ki | 11 | — | |
DLWMVUDMPMKGEE
|
6.5 | Ki | 24 | — | |
JCFJQIHDZHHMQT
|
6.5 | Ki | 42 | — | |
MMFBBQQGBVPLQQ
|
6.5 | Ki | 13 | — | |
OLVBAUVSICCWEJ
|
6.5 | Ki | 39 | — | |
XMGFTZYNTYNOOJ
|
6.5 | Ki | 10 | — |