Target Details
| UniProt AC | P08922 |
|---|---|
| Gene Symbol | ROS1 |
| Protein Name | Proto-oncogene tyrosine-protein kinase ROS |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 263
- Clinical molecules 18
- Avg pChEMBL 7.6
Associated Diseases (1)
Active Molecules (263)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HAYYBYPASCDWEQ
|
8.2 | IC50 | 47 | — | |
JFJBQYDTDVUFOI
|
8.2 | IC50 | 3 | — | |
AIQDZMUPVYDVLB
|
8.1 | Ki | 48 | — | |
GPAQVHTXRUBATF
|
8.1 | IC50 | 2 | — | |
VALNJAQHJPYEAK
|
8.1 | IC50 | 3 | — | |
XKFTZKGMDDZMJI
|
8.1 | Ki | 56 | — | |
IROGUEMYXINLOZ
|
8.1 | IC50 | 3 | — | |
ARFSIMCXZSKBGL
|
8.1 | IC50 | 3 | — | |
MMZVTNYPOASLID
|
8.1 | IC50 | 3 | — | |
MPLLJMUCCXFTPL
|
8.1 | IC50 | 3 | — | |
NRFLPOVNIIJIDX
|
8.1 | IC50 | 3 | — | |
NVTUEJKEIISOPJ
|
8.1 | IC50 | 3 | — | |
NWDUSAJTSMCLKW
|
8.1 | IC50 | 3 | — | |
RONLQWJKAFWDOO
|
8.1 | IC50 | 3 | — | |
SUZGZTADNRRPLU
|
8.1 | IC50 | 3 | — | |
YNXUIZMRPVCJTM
|
8.1 | IC50 | 3 | — | |
MGGBYMDAPCCKCT
|
8.1 | IC50 | 23 | — | |
JPUUSJUGUJODFK
|
8.0 | IC50 | 2 | — | |
KHNKMLQHLHWWSI
|
8.0 | IC50 | 3 | — | |
RQZIXOOARXBNHW
|
8.0 | IC50 | 2 | — | |
UOIPIFGVZNDCCW
|
8.0 | IC50 | 2 | — | |
MZDKLVOWGIOKTN
|
7.9 | Ki | 80 | — | |
ZHOXAGNPCZTRBN
|
7.9 | Kd | 20 | — | |
RACYTTCRBPEXAP
|
7.9 | IC50 | 2 | — | |
SEJGTFPOEJWEGG
|
7.8 | Kd | 149 | — | |
HZTYDQRUAWIZRE
|
7.8 | Kd | 40 | Yes | |
CXQHYVUVSFXTMY
|
7.8 | Ki | 154 | — | |
SQPURFIALRFCBJ
|
7.7 | IC50 | 2 | — | |
DBXGGXLBTWZXBB
|
7.7 | Ki | 39 | — | |
UOVCGJXDGOGOCZ
|
7.7 | Ki | 59 | — | |
NRFMLFPXDKIQBF
|
7.7 | Kd | 8 | — | |
MULNSLQVKKUPJN
|
7.6 | Ki | 41 | — | |
UQJQNZHGEVLHST
|
7.6 | Ki | 15 | — | |
YEHCNYAQEBQCCS
|
7.6 | Ki | 74 | — | |
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
BNXYQBUYYXJKBW
|
7.6 | IC50 | 3 | — | |
JXPQCRCHIRKWDH
|
7.6 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
7.5 | Kd | 220 | — | |
NCZKBNXMSRBQNT
|
7.5 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.5 | Kd | 213 | — | |
RPGBQFNDFPEOON
|
7.5 | Ki | 22 | — | |
RYYNGWLOYLRZLK
|
7.5 | Ki | 104 | — | |
ZVWRFVCNQOECJS
|
7.5 | Ki | 71 | — | |
BLYRPGBSIKAIAU
|
7.4 | IC50 | 24 | Yes | |
MICOMLRETSSUOK
|
7.4 | IC50 | 3 | — | |
MIKAKZKNMYZLDX
|
7.3 | Ki | 42 | — | |
UQKLTKAHTNLXPA
|
7.2 | IC50 | 5 | — | |
PBBXBBSBAJKYLC
|
7.2 | Kd | 3 | — | |
CZQVOIDVDAVDFW
|
7.2 | Ki | 18 | — | |
HCNIBOQWDVOZKF
|
7.2 | Ki | 26 | — |