Target Details
| UniProt AC | P08922 |
|---|---|
| Gene Symbol | ROS1 |
| Protein Name | Proto-oncogene tyrosine-protein kinase ROS |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 263
- Clinical molecules 18
- Avg pChEMBL 7.6
Associated Diseases (1)
Active Molecules (263)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZUSOUYHYDDCGIC
|
8.6 | IC50 | 4 | — | |
LVMSBBICHCLRMS
|
8.6 | IC50 | 2 | — | |
WHVFDYQCAMPLMS
|
8.6 | Ki | 20 | Yes | |
IJKDASOGZQSXII
|
8.6 | IC50 | 2 | — | |
OEBIHOVSAMBXIB
|
8.6 | IC50 | 5 | — | |
WQLHYGLQUAJXEC
|
8.6 | IC50 | 2 | — | |
DOWWFGLYJNBUSG
|
8.6 | IC50 | 4 | — | |
FGRVKMDGFGXLDX
|
8.6 | IC50 | 5 | — | |
GCAJYDBNZMKHTH
|
8.6 | IC50 | 3 | — | |
HKTKCWHAQWAVOW
|
8.6 | IC50 | 5 | — | |
LTPMGUPHSVPNRT
|
8.6 | IC50 | 3 | — | |
NXPHBBCDRJWBHG
|
8.6 | IC50 | 3 | — | |
OUBJSHKDVMRZQJ
|
8.6 | IC50 | 5 | — | |
POXSFRWIBWNONT
|
8.6 | IC50 | 3 | — | |
QRMNFHGVKRGQBQ
|
8.6 | IC50 | 3 | — | |
RLHGMHDDJDTUOF
|
8.6 | IC50 | 3 | — | |
SCHLJLHHIALWBK
|
8.6 | IC50 | 5 | — | |
SXRLSRMWBAVNFG
|
8.6 | IC50 | 3 | — | |
VROSTPWCFHKXPW
|
8.6 | IC50 | 4 | — | |
WHODNMAIHAPRJL
|
8.6 | IC50 | 3 | — | |
WJAQYAUNJKXATP
|
8.6 | IC50 | 3 | — | |
XNLDXKJZCGYOAU
|
8.6 | IC50 | 5 | — | |
GZSOMRIONXRGEX
|
8.5 | IC50 | 4 | — | |
JTLQSWMRBFBYEA
|
8.5 | IC50 | 2 | — | |
XOOAAYRIVATZNM
|
8.5 | Ki | 55 | — | |
PKMJFPBKTISKAX
|
8.5 | IC50 | 3 | — | |
AJHJEQWEJUXGIF
|
8.5 | IC50 | 4 | — | |
SVUZWKKSPKPLEO
|
8.4 | IC50 | 2 | — | |
AOXIGKGAMMGXCX
|
8.4 | IC50 | 2 | — | |
SNYQSPGQFDKITH
|
8.4 | IC50 | 3 | — | |
XKZINYYXWJEYEL
|
8.4 | Ki | 37 | — | |
QOEFDQQUMQBVOB
|
8.4 | IC50 | 2 | — | |
BAKDYDIANXRUHQ
|
8.4 | IC50 | 3 | — | |
CMVRVFZXCSVCKY
|
8.3 | IC50 | 2 | — | |
YGYGMNYVMRIARK
|
8.3 | IC50 | 3 | — | |
LVLFSSZNAIKYCD
|
8.3 | IC50 | 19 | — | |
PEKQRSRFUKHNAB
|
8.3 | IC50 | 2 | — | |
SRWSLWJKGRZRMC
|
8.3 | Kd | 4 | — | |
KQYVFELJSCVCND
|
8.3 | IC50 | 4 | — | |
NHEOMGKMIVQQIX
|
8.3 | IC50 | 4 | — | |
UYJNQQDJUOUFQJ
|
8.3 | Ki | 68 | — | |
WPHKIQPVPYJNAX
|
8.3 | Ki | 81 | — | |
ZWVZORIKUNOTCS
|
8.3 | Ki | 69 | — | |
JWHAROIQSCGUPR
|
8.3 | IC50 | 2 | — | |
KUFBKQQDUMDVPE
|
8.3 | IC50 | 2 | — | |
ATUIHXRIJCYLPA
|
8.3 | IC50 | 4 | — | |
GYQWOGHOBIBGDV
|
8.2 | IC50 | 4 | — | |
JZTOUVBEZONDKA
|
8.2 | Ki | 80 | — | |
KTEIFNKAUNYNJU
|
8.2 | IC50 | 114 | — | |
XTOSJDBUWRFEGO
|
8.2 | IC50 | 3 | — |