Target Details
| UniProt AC | P08922 |
|---|---|
| Gene Symbol | ROS1 |
| Protein Name | Proto-oncogene tyrosine-protein kinase ROS |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 263
- Clinical molecules 18
- Avg pChEMBL 7.6
Associated Diseases (1)
Active Molecules (263)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DIXMBHMNEHPFCX
|
10.7 | Ki | 12 | — | |
HKSZLNNOFSGOKW
|
10.2 | IC50 | 49 | Yes | |
FIKPXCOQUIZNHB
|
9.8 | IC50 | 9 | — | |
VXYZCOCRVAQWBG
|
9.7 | Ki | 15 | — | |
HKSZLNNOFSGOKW
|
9.7 | IC50 | 408 | — | |
WUOOWFKJQHKXHK
|
9.7 | IC50 | 4 | — | |
LRJJEMRURFIKDD
|
9.7 | IC50 | 6 | — | |
IIXWYSCJSQVBQM
|
9.6 | Ki | 18 | — | |
VPTLPKOEIZQIAS
|
9.5 | IC50 | 4 | — | |
FOLXFWBVNHRGIV
|
9.5 | IC50 | 6 | — | |
AKARKHHDGYZKIF
|
9.5 | IC50 | 5 | — | |
HKSZLNNOFSGOKW
|
9.5 | IC50 | 118 | — | |
VGEDWONGQUXJQA
|
9.5 | IC50 | 7 | — | |
OWRXHGAFWZFFCW
|
9.4 | Ki | 113 | — | |
SSPYHBZSDDTSFN
|
9.4 | IC50 | 9 | — | |
DPMQHTABGLRCQK
|
9.4 | IC50 | 5 | — | |
KZNWRBSYSUFFOG
|
9.3 | IC50 | 2 | — | |
GDVDELGPSHNWGV
|
9.3 | IC50 | 4 | — | |
LTTXNEAUXULKJC
|
9.2 | IC50 | 2 | — | |
BNPMMVDYMYENIM
|
9.2 | IC50 | 4 | — | |
TTWJGJUDRLYONZ
|
9.1 | Kd | 6 | — | |
UQWDXRWKSYDDTE
|
9.1 | IC50 | 2 | — | |
SXTUUDANYSHGTB
|
9.1 | IC50 | 2 | — | |
NFVNVIQUEXSEFR
|
9.1 | IC50 | 4 | — | |
NFUNPZHOYQJPEH
|
9.1 | IC50 | 2 | — | |
IXBQYIJFDYAVJA
|
9.0 | IC50 | 2 | — | |
WTHYAPGHJBPUJT
|
9.0 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
9.0 | IC50 | 231 | Yes | |
TVUWQDLBEOZVOU
|
9.0 | Ki | 41 | — | |
UMZFBMAHLWQSBF
|
9.0 | IC50 | 4 | — | |
MYBIYOGYGXIDJG
|
9.0 | IC50 | 2 | — | |
DTCJOPXFZUJREL
|
8.9 | IC50 | 2 | — | |
PWCNVYNJXOVGLO
|
8.9 | IC50 | 4 | — | |
SHRNMJSKKQHLKT
|
8.9 | IC50 | 4 | — | |
OHIKHZFSGQMGGD
|
8.9 | IC50 | 5 | — | |
KTEIFNKAUNYNJU
|
8.8 | Ki | 48 | — | |
CWQBEWYRKVPJHU
|
8.8 | IC50 | 2 | — | |
JZCIRSHLQAWPRJ
|
8.8 | IC50 | 2 | — | |
YISMQBFJYDFMAL
|
8.8 | IC50 | 46 | — | |
STKCTXOVMCUJSB
|
8.7 | IC50 | 4 | — | |
AILRADAXUVEEIR
|
8.7 | IC50 | 75 | — | |
IEBZBPYYZNDTMO
|
8.7 | IC50 | 4 | — | |
MAKLQLGGXQPLRV
|
8.7 | IC50 | 2 | — | |
OVDSPTSBIQCAIN
|
8.7 | IC50 | 7 | — | |
CQRRHOGDBIREMX
|
8.7 | IC50 | 2 | — | |
GDRLJBDXWDATLA
|
8.7 | IC50 | 13 | — | |
RBXYGQNZRVPDNB
|
8.7 | Ki | 34 | — | |
VERWOWGGCGHDQE
|
8.7 | IC50 | 23 | — | |
DIWRJVJHXXZINL
|
8.6 | IC50 | 4 | — | |
IVWSMDDTFYCVFZ
|
8.6 | IC50 | 2 | — |