Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
CPNQDPLKZHXMSB 7.0 Ki 6
LCPAFKZCFFLTPB 7.0 Ki 3
MHEKDRNEOKTABI 7.0 IC50 2
MNMDMCKHXVHLAW 7.0 Ki 3
NSXUBFCOCMDGJL 7.0 Ki 6
UVOCSZKGWJOKNN 7.0 Ki 11
SGVJKODGLNRNLW 7.0 Ki 18
WIKYUJGCLQQFNW 7.0 IC50 23 Yes
GLMXKJUUSZJNIE 7.0 Ki 2
WPNJAUFVNXKLIM 7.0 Ki 4
GPEOXJGBWGMANI 7.0 IC50 2
QNKGTIWNFNPEJL 7.0 Ki 11
RWVUEZAROXKXRT 7.0 IC50 11
VGIYMYGMVXPMKV 7.0 Kd 3
XETGFITVYCWVGB 7.0 Ki 6
XJARKGGVDJGJMK 7.0 IC50 2
SYPINLPWMTYMEC 7.0 Ki 3
MBYSTKNEMJZSIK 6.9 Ki 6
MOWCGUQGNSAZSR 6.9 IC50 2
ALTKABGEMCJWJH 6.9 Ki 15
APNJYYQXBHETAR 6.9 Ki 3
CVKQUGPVDVFRAT 6.9 Ki 4
DHSSDEDRBUKTQY 6.9 Ki 6
QZUDBNBUXVUHMW 6.9 Ki 39 Yes
RGPTYLNPCNVHNC 6.9 Ki 8
UFVSFWQCSISIPB 6.9 Ki 3
LQEATNFJCMVKAC 6.9 Ki 14
ZMDCNVSZNFXVKI 6.9 Ki 3
ACTVOFFLDWZANE 6.9 Ki 9
ACTVOFFLDWZANE 6.9 Ki 9
QKDDJDBFONZGBW 6.9 Ki 5
QLOOWOVVZLBYHU 6.9 Ki 7
TVDZYHOTHAFPBR 6.9 Ki 2
YFPXOLILPOTYIP 6.9 Ki 5
GPEOXJGBWGMANI 6.9 IC50 3
HZPGVFKYDDQWIZ 6.9 IC50 4
IESRGXWBZDJPLC 6.9 IC50 2
NJWKXGIQDOFDKH 6.9 IC50 3
WEGLOYDTDILXDA 6.9 Ki 22
AFRRMVBYOMNLHN 6.9 Ki 3
VLMCHIMKCURVRR 6.9 Ki 3
AFWQDDUMQAQVSC 6.9 Ki 3
HIJHJEWMVKEUOP 6.9 Ki 3
BKDDSROSFZKQTN 6.8 IC50 2
BQJCRHHNABKAKU 6.8 Ki 4
JYEPTVGXWUQMKF 6.8 Ki 2
YZDFADGMVOSVIX 6.8 Ki 16
NEUSVAOJNUQRTM 6.8 IC50 13 Yes
XAFOTAKURAOBIE 6.8 Ki 6
CJAWPFJGFFNXQI 6.8 Ki 4
2D structure