Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
DAEHQHNTEAMXQC 7.1 Ki 3
HVCWUSZDSFHZDW 7.1 Ki 3
NMSAVNXFCXMJJY 7.1 Ki 2
ODGBUUUVMLDZBP 7.1 Ki 7
CEUORZQYGODEFX 7.1 Ki 31
DFZXRUBHUWNVAN 7.1 Ki 3
ICROYPJYNVAMQF 7.1 Ki 3
QFKQUMBUFVKQBH 7.1 Ki 5
RIMQFOFQYZBTDB 7.1 Ki 3
FASDKYOPVNHBLU 7.1 Ki 9
NFSIDEIKDWWMOX 7.1 Ki 2
PCMKFHUKCPUDQK 7.1 IC50 2
RVIXAJHMKWFIKC 7.1 Ki 3
HLVQBOYEHQRWHG 7.1 Ki 5
OTXMFMMMNBKXQC 7.1 Ki 4
OYOGQACTFBHTOD 7.1 Ki 3
ZFYOCHWWKWULRT 7.1 Ki 3
KLBQZWRITKRQQV 7.1 IC50 25 Yes
MZDQVKPPFWIZIL 7.1 Ki 5
NMSAVNXFCXMJJY 7.1 Ki 3
RREJZKOLYMUBNO 7.1 Ki 5
XRJGWSMTLAFHBN 7.1 Ki 21
JWPAYBAIIARWMG 7.1 Ki 19
OHLOMHGVALXPJP 7.1 Ki 3
PANBMHHKBRMYAL 7.1 Ki 5
YQBKUZKHVPTFOO 7.1 Ki 2
XPKLCTLEXRSJEM 7.1 IC50 2
ZUXABONWMNSFBN 7.1 Ki 29
MQZXNJVAUSWZRL 7.1 Ki 3
URKOMYMAXPYINW 7.1 Ki 27 Yes
VPDYOWAJRMPOEI 7.1 Ki 3
KRFMDKUGQLNZKI 7.0 Ki 3
OQDPVLVUJFGPGQ 7.0 Ki 9
OGOLMGZJNRNULQ 7.0 Ki 3
QPAIAAWBFFTOPZ 7.0 Ki 2
DAKGDRVNCPHAPY 7.0 Ki 5
OABROWXKGQFLDH 7.0 Ki 3
RNPCOHCWKNMBRI 7.0 Ki 3
CJGNMVAAMQAWEF 7.0 Ki 16
KSQOPRCDYFOHET 7.0 Ki 4
MEKSQRMXWZHFIP 7.0 Ki 13
OLPQNRLJYOGSGV 7.0 Ki 6
PSVIJGBMZYPVMJ 7.0 Ki 3
UEZSUAXJWCMWEK 7.0 Kd 3
CYJMDICCNHFYPK 7.0 IC50 2
DYQQPAOLMYPZKE 7.0 Ki 2
IHCKEJIXIYLTFT 7.0 Ki 2
UULIGRNKXHCLQN 7.0 IC50 2
UULIGRNKXHCLQN 7.0 IC50 2
XGMNRALXOWECNG 7.0 Ki 3
2D structure