Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
PXPKAXRRJYZLDN 7.3 Ki 3
SNBRKKJCZXXNNL 7.3 Ki 3
UGUPGQUFTPDBTH 7.3 IC50 2
CJFOJUCLYBZSAN 7.3 Ki 3
OGOLMGZJNRNULQ 7.3 Ki 4
YGIWTZGEYHABOR 7.3 Ki 6
KJTFLBJQHBFQAF 7.3 Ki 5
XBWFPEVESQMIBM 7.3 Ki 3
CKZOGIXOGHVXNW 7.3 Ki 3
NFKNRFTZWQGNTI 7.3 Ki 4
WIQCERUTOBWUOL 7.3 Ki 3
FLAHEXULHVZYHT 7.3 Ki 3
OITKDPXYSUWTOJ 7.3 Ki 3
GPPWMDRIVISCNC 7.3 Ki 3
MNMDMCKHXVHLAW 7.3 Ki 4
PFTFJTOQCWYCNM 7.3 Ki 3
NYGANYRUZQPPGP 7.3 Ki 5
QNWVOPOAKHMIHV 7.3 Ki 3
UZRVBSAZMGMVTH 7.3 Ki 3
OHRDRIOXKSBXGK 7.2 Kd 6
AJWTXSLKVJNYAB 7.2 Ki 3
JJQLRTKUCLCIPR 7.2 IC50 3
LDCMGLYXOOMRFQ 7.2 IC50 3
MCAGSCISRRGDGQ 7.2 Ki 3
MNMDMCKHXVHLAW 7.2 Ki 4
RCMYMJSBSVKJNP 7.2 IC50 2
SQPFWLZXWYXMCI 7.2 Ki 3
XBBHVMXFPPVGMX 7.2 Ki 6
YAORIDZYZDUZCM 7.2 Ki 5
BXGRLXRXUOGKTC 7.2 IC50 2
NMSAVNXFCXMJJY 7.2 Ki 3
XFYDIVBRZNQMJC 7.2 Ki 2
PPJRQXMDFSRWFH 7.2 Ki 3
RFTNZWFCHDUSMZ 7.2 IC50 2
YVENIGOVHPMTDH 7.2 Ki 23
ZVVQFUFKMNLNCB 7.2 Ki 6
NGEQXHFDGLOZSS 7.2 Ki 2
NREVCQNJBZJFTB 7.2 Ki 2
NTSMKZTVZAMTDB 7.2 Ki 8
PVKUNRLEOHFACD 7.2 Ki 3
BSOLCASXROXPRZ 7.2 Ki 9
OGHNVEJMJSYVRP 7.2 IC50 18
SNKCREOVGWDJDI 7.2 Ki 3
AOQYWVCOSJELMS 7.2 Ki 3
MRSWPVWIMKYKPA 7.2 Ki 3
HJACXCAXDLNLEL 7.2 Ki 3
INJOMKTZOLKMBF 7.2 Ki 6
FTXAKSJEBVGKHR 7.2 IC50 2
YEHCICAEULNIGD 7.2 Ki 20
BSOLCASXROXPRZ 7.1 Ki 9
2D structure