Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
UFIMBHYPDHTMKA 7.5 Ki 4
ARHDCTCZSSOSFG 7.5 Ki 3
DRHKJLXJIQTDTD 7.5 Ki 9
PMXMIIMHBWHSKN 7.5 Ki 19
AEWIKTWIKIWVNJ 7.5 Ki 2
BAAUEDJUTZLMAN 7.5 Ki 6
PIAONGWBRPZERV 7.5 Ki 3
UGTJLUOFSLGNDT 7.5 IC50 3
FZQJYKJEUSSHNW 7.5 Ki 3
NEEHDLNCAAFDSD 7.5 Ki 3
OXGCVSXSSWZTMU 7.5 Ki 3
VRYMTAVOXVTQEF 7.5 Kd 6
CHKGJSUYXRACOM 7.5 Ki 3
IYLGKCYRBQLWIN 7.5 Ki 3
ZTBWRKAKTUWRSC 7.5 Ki 3
KZRCWZJRCYMXFF 7.5 IC50 2
LFMHROBTZOFVNB 7.5 Ki 3
SWMRFMZFBGUQMK 7.5 Ki 2
WSSHHAWIZNWBLH 7.5 Ki 3
LGTDYALRCIBCMI 7.5 Ki 3
CQXADFVORZEARL 7.4 Ki 4
LAEXASCTDHUYIT 7.4 Kd 3
NKVMZSSSOMIEIA 7.4 Ki 6
SEKAQUSPSDPIAN 7.4 Ki 4
SGUAFYQXFOLMHL 7.4 Kd 11
HUCJFAOMUPXHDK 7.4 Ki 8
VJQWCCBDYLTRPZ 7.4 Ki 3
YVSAGYHRJDVYHG 7.4 Ki 3
LJRFIWIVFLBBPS 7.4 Kd 6
NYGHGTMKALXFIA 7.4 Ki 4
QELYRGGNEIAOKD 7.4 Ki 2
XGMNRALXOWECNG 7.4 Ki 3
OSJJYEUEJRVVOD 7.4 IC50 17 Yes
WBGSURPVIDDDHF 7.4 Ki 3
FVORBSYXXHDBGZ 7.4 Ki 3
RKQFKAILJGXGRP 7.4 Ki 3
RONZAEMNMFQXRA 7.4 IC50 9 Yes
SEKAQUSPSDPIAN 7.4 Ki 4
ZHDIISZEXUGDAJ 7.4 Ki 6
ACQBHJXEAYTHCY 7.4 Ki 5
PKXHLBVPUHXZNH 7.4 Ki 3
IAIZHDGEGFGNMO 7.3 Ki 3
QYCJTZDZQXSXSC 7.3 Ki 3
SEKAQUSPSDPIAN 7.3 Ki 4
IAIZHDGEGFGNMO 7.3 Ki 3
PNISAWOKGCKONH 7.3 Ki 4
RWDJYHMGMOOTRK 7.3 Ki 3
VAYOSLLFUXYJDT 7.3 Ki 19
LDCMGLYXOOMRFQ 7.3 IC50 2
PJHALOKEQHBBKK 7.3 Ki 3
2D structure