Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
UDQDKOIZHDPWGR 7.8 Ki 3
DZSQSLQSMKNVBV 7.8 Ki 4
UEQUQVLFIPOEMF 7.8 Ki 13
RCLSMBSYDRCUSB 7.8 Ki 3
TVTNBOZUNDIPJR 7.8 Ki 5
YAYASQTZIRSRFB 7.8 Ki 3
LJLYHROZJUTILK 7.8 Ki 3
UCAIEVHKDLMIFL 7.8 Ki 4
BCCMUPQZPVRDCD 7.7 Ki 6
BQXXXVQLOOIBPN 7.7 Ki 3
NATLAODAVOGBDD 7.7 Ki 3
UEQUQVLFIPOEMF 7.7 IC50 21 Yes
KKJVPLDLUKVODK 7.7 Ki 3
MKDJCTAYFLKGEM 7.7 Ki 3
HCMWMLSNHRNVSJ 7.7 Ki 3
SPMYVDNOOYXROZ 7.7 Ki 3
CNIIGCLFLJGOGP 7.7 Ki 4
GJSURZIOUXUGAL 7.7 Ki 9
QYCJTZDZQXSXSC 7.7 Ki 4
RYUJZKYTNJACIJ 7.7 IC50 3
WFPUBEDBBOGGIQ 7.7 Ki 4
YEPGXJIOCYXZAI 7.7 Ki 3
AQDOXXILINNVJB 7.7 Ki 3
ASMAFSDTDIBMNU 7.7 Ki 4
GEBHRBBICJPJRU 7.7 Ki 3
XMXHEBAFVSFQEX 7.7 Ki 17
AUVVAXYIELKVAI 7.6 IC50 10
BGPHEWUAKSHOBD 7.6 Ki 3
NFGYJBCMYUYKCI 7.6 Ki 4
QYCJTZDZQXSXSC 7.6 Ki 4
WZOMJNATDSYQHS 7.6 Ki 3
ONSCHPQYHGOIQX 7.6 Ki 6
RUFDXBQFEDFKDE 7.6 Ki 3
WKXSXFYQPCWZOS 7.6 Ki 6
ZBEZMDBAFCFGAT 7.6 Ki 6
LYKMMUBOEFYJQG 7.6 Kd 6
NGYGSYPEYBVPQK 7.6 Ki 3
RLKWQKZPCMICPS 7.6 Ki 3
WDZVGELJXXEGPV 7.6 IC50 8
LAMFPOWZDAOQTK 7.6 Ki 3
WYFPZXUWZCKNMJ 7.6 Ki 3
YWALOGYVALOLTL 7.6 Ki 3
BFSPTAYUYXLBEU 7.6 Ki 3
MDFFTELFADBPIZ 7.6 Ki 4
MPCNSEQVVHOHGO 7.6 Ki 3
SJTUPIJPFNBFHK 7.6 Ki 3
XGMNRALXOWECNG 7.6 Ki 3
IBNWNWKMISLVQT 7.5 Ki 8
IPQYPIRIGUBUAF 7.5 Ki 3
JFKKLIJAJCMWRM 7.5 Ki 8
2D structure