Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
HGEYJZMMUGWEOT 8.2 Ki 17
IAHLXXAKFXOKST 8.2 Ki 3
CETMNKCDAHCKRC 8.2 Ki 3
GUYATMODRNZQDL 8.2 Ki 6
NEQHKSNFFVEGHN 8.2 Ki 6
RTHCYVBBDHJXIQ 8.2 Ki 15 Yes
RTHCYVBBDHJXIQ 8.2 Ki 15
CUHVIMMYOGQXCV 8.2 Ki 7
HAEPGZUGYMHCJE 8.2 Kd 3
YYTGOWDNUUXBGS 8.2 Ki 5
HAEPGZUGYMHCJE 8.2 Kd 3
KXSUAWAUCNFBQJ 8.1 Ki 3
NWUCPBLQECHRFK 8.1 IC50 3
NWUCPBLQECHRFK 8.1 IC50 3
WLQWOUULTDRZTQ 8.1 Ki 3
HPMRFMKYPGXPEP 8.1 Ki 10
VDDKWLCHDOJXJM 8.1 Ki 3
XSOUHEXVEOQRKJ 8.1 Ki 14
NADZGFHXOOQKNN 8.1 Ki 3
UEZSUAXJWCMWEK 8.1 Kd 3
GHIKYGQWBRHEGU 8.1 Ki 2
WYWIFABBXFUGLM 8.1 Ki 17
WZOMJNATDSYQHS 8.1 Ki 3
XXQLSAWUSXSJTK 8.1 Ki 6
CVKQUGPVDVFRAT 8.1 Ki 3
KOMMMRWKUHRBSF 8.0 Ki 3
RSRUDTPYRBLHEO 8.0 Ki 6
PGOVKWAJCVAZNG 8.0 Ki 3
XDAIWLKBRMSRTM 8.0 Ki 2
HSSBMQXDKGERBI 8.0 Ki 4
BEAKKNUWBXQLLR 8.0 Ki 2
KENQBAJESGJICP 8.0 IC50 2
KKLYBLFGKSXYJZ 8.0 IC50 4
RAPZEAPATHNIPO 8.0 Ki 28 Yes
RHPCETHLGGFAQB 8.0 Ki 9
VSWBSWWIRNCQIJ 8.0 Ki 23
JVGBTTIJPBFLTE 8.0 Ki 16
WUTIBZPSZGYSGD 8.0 Ki 3
AWPNMWRTPSQMFC 7.9 Ki 2
HSSBMQXDKGERBI 7.9 Ki 4
JWAAXMLRAVOKBQ 7.9 Ki 3
KORNTPPJEAJQIU 7.9 Ki 17
MOJPEWKNYNURQQ 7.9 Ki 2
RWMIVZPIQPHMSK 7.9 Ki 3
OZVBMTJYIDMWIL 7.9 Ki 20
NUMRIDYCRYHYHT 7.9 Ki 3
VNSOQQZNVNIEMP 7.9 Kd 6
KSMAGQUYOIHWFS 7.8 Ki 3
OOYTZYZXCMCMSZ 7.8 Ki 3
RATZLMXRALDSJW 7.8 Ki 4
2D structure