Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
HSWPZIDYAHLZDD 8.7 Ki 3
VMLJCXYBTLCGDU 8.7 Ki 3
IRIQHWJBJQBIEB 8.7 Ki 3
QZUXRMOPAGPTIY 8.7 Ki 4
WGLYZLZIIJTKAG 8.7 IC50 4
FXNNPMSELIMMHU 8.6 Ki 4
MHPMXTGKTXJIDI 8.6 Ki 6
WZOMJNATDSYQHS 8.6 Ki 6
XYLJNLCSTIOKRM 8.6 Ki 4
MNHDKMDLOJSCGN 8.6 Ki 23
BLAVUEWHVKGIIM 8.5 Ki 3
LEHLBTBBMZYRBK 8.5 Ki 3
WEXLHWFGOZCTNY 8.5 Ki 3
HQDWMIAYEGTBSF 8.5 Ki 3
WDSZUSABLKNHCZ 8.5 Ki 3
WDSZUSABLKNHCZ 8.5 Ki 4
CARQBUHFBAORAB 8.5 Ki 3
ASHFKBMVCDTQQO 8.5 Ki 4
IDRYZRZTCSBDSQ 8.5 IC50 2
UCNOTTVNPRSTFW 8.5 Ki 8 Yes
GYSZUJHYXCZAKI 8.5 Kd 7
MBPZQLMDDBIIGZ 8.5 IC50 3
RJGDAIXCXQIWEK 8.4 IC50 3
UJYGDMFEEDNVBF 8.4 IC50 12
IEJXVRYNEISIKR 8.4 Ki 6
IXRPDYSTGHYEBR 8.4 Ki 4
WUSIUKLVFNJEHL 8.4 Ki 3
AUMIZIKCBYPWJM 8.4 Ki 3
IOEIAXGHDJMROV 8.4 Ki 2
MRBDMNSDAVCSSF 8.4 Ki 10
KSMAGQUYOIHWFS 8.4 Ki 4
UFWIBTONFRDIAS 8.3 Ki 3
VSRXHPMNIVBYAT 8.3 Ki 2
DGXYDPJRLWCWFV 8.3 Ki 3
YRVKJIDCHIEELY 8.3 Ki 6
HAIKGHUWKLUYNG 8.3 Ki 2
YDOTUXAWKBPQJW 8.3 IC50 13
AZADEQYOIWOMER 8.3 Ki 2
CUHVIMMYOGQXCV 8.3 Ki 6
XHLHZPFSBCZVEA 8.3 Ki 6
XHLHZPFSBCZVEA 8.3 Ki 3
FAFGGANFZMERDR 8.3 Ki 3
NJTFNKZJGXSOMJ 8.3 Ki 3
RQEBRILFCMJWAD 8.3 Ki 2
DAIRUBYTBODIKT 8.3 Ki 3
SGOFAUSEYBZKDQ 8.2 Ki 2
HBMJQYDGBNSZMC 8.2 Ki 4
WNCGPEYSCDVJNB 8.2 Ki 3
JDFLCCTUDMVCCS 8.2 Ki 2
GNQMAWAOPDTCCX 8.2 Ki 3
2D structure