Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
YMYZKGIHGMHZDL 9.2 Ki 5
UDURNHDRCUMUOV 9.2 IC50 4
DISVZQSFAXIOLP 9.2 Ki 3
BKRGVLQUQGGVSM 9.1 Ki 26 Yes
FJABWASNVHOPLU 9.1 Ki 3
JWYUBODPEUBFLH 9.1 Ki 3
JWYUBODPEUBFLH 9.1 Ki 11
HOKCXDCTKLQEJE 9.1 Ki 3
LQKQCQKZRUYZOI 9.1 Ki 4
COPXFRMTXFPQKE 9.1 Ki 3
HNRZWHPQDGUUSO 9.1 IC50 4
MUUSOYWTPTTZII 9.1 Ki 3
MUUSOYWTPTTZII 9.1 Ki 3
QHCZSHHKZDDCEC 9.1 Ki 3
HQGWKNGAKBPTBX 9.0 Ki 3
DMVFXOFRGGGXKJ 9.0 Ki 2
FDVZSKDDSYLYNX 9.0 Kd 4
OLAGLCHGSUYVBF 9.0 Ki 3
PYXVPLGVUNHGEJ 9.0 Ki 3
ZMOPTLXEYOVARP 9.0 Ki 14 Yes
LUZRJRNZXALNLM 9.0 Ki 20
IPLOTOHAAAUTMK 9.0 Ki 3
JCJVFLLBDXJJPW 9.0 Ki 3
JWXMKFUDAOLJCY 9.0 Ki 4
JRMVEEDZCPVFFK 8.9 IC50 3
CAIGGWCQMXMLII 8.9 Ki 3
OSJZLDGTMVBIRV 8.9 Ki 6
DEQITUUQPICUMR 8.9 IC50 13
UVEKKXRFQCNLQE 8.9 Ki 4
LLFVSLMMRPXQFK 8.9 Ki 3
RJLMZCSOGDTDNJ 8.9 Ki 3
XCGSFFUVFURLIX 8.9 IC50 17
VKABNRMTNPWHBD 8.9 Ki 3
BSOFNSGMVOMVLM 8.8 Ki 3
YMYZKGIHGMHZDL 8.8 Ki 3
MGQIWQQQIZXANT 8.8 Ki 3
FYLKUCQQWYKEOG 8.8 Ki 4
HSRPTPAPMBHRRJ 8.8 IC50 5
WFPDOLGWGNFUFR 8.8 IC50 3
GHPKBFZQNLPFFZ 8.8 Ki 3
GHPKBFZQNLPFFZ 8.8 Ki 3
LWSVCEUUPRLOSZ 8.8 Ki 3
JPNJJWFOEQLLSP 8.8 Ki 3
KSQAWHREGPMSBF 8.8 Ki 3
NDFYRGCPDAFQDG 8.8 Ki 2
VUQFQRNHGGYQGK 8.8 Ki 3
JMXRRARDLWHYJN 8.8 IC50 4
RVRPAIWBGBVSKB 8.8 Ki 3
SATXLDNXPGMNQI 8.7 Ki 3
UAHLUVNKSWGJEK 8.7 Ki 3
2D structure