Target Details
| UniProt AC | P08913 |
|---|---|
| Gene Symbol | ADRA2A |
| Protein Name | Alpha-2A adrenergic receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 761
- Clinical molecules 54
- Avg pChEMBL 7.3
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (761)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GKTQBPYMIGXPKG
|
6.0 | Ki | 21 | Yes | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
PNVNVHUZROJLTJ
|
6.0 | Ki | 6 | — | |
SLGLZEJKMBCODK
|
6.0 | Ki | 4 | — | |
SOPASBFWKHVOQL
|
6.0 | Ki | 3 | — | |
TZJUVVIWVWFLCD
|
6.0 | IC50 | 8 | Yes | |
VHGCDTVCOLNTBX
|
6.0 | Ki | 19 | — | |
WGHJKYWWSVIRLL
|
6.0 | IC50 | 7 | — | |
XNHVIEKFPXTSAV
|
6.0 | Ki | 3 | — | |
ZDDQYDGPVSLKGX
|
6.0 | Kd | 6 | — | |
ZEUITGRIYCTCEM
|
6.0 | Ki | 12 | — |