Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
VCKUSRYTPJJLNI 6.3 Ki 6
ZAKQYSXDZKMEJJ 6.3 Ki 2
BYPMJBXPNZMNQD 6.2 Ki 18
IOIMNYMJVKCZNT 6.2 Ki 3
VSWYSDPXUHVQCG 6.2 Ki 11
AIMNRLCNWYRUPJ 6.2 IC50 4 Yes
GKIRPKYJQBWNGO 6.2 IC50 20 Yes
INNDGUNGHHCVFO 6.2 IC50 2
IZBNNCFOBMGTQX 6.2 Ki 5
NTJQREUGJKIARY 6.2 Ki 7
OJJDBXUPMILXPO 6.2 Ki 3
QOYHHIBFXOOADH 6.2 Ki 16
SGTNSNPWRIOYBX 6.2 IC50 19
SPIJYUMJUFXBOQ 6.2 Ki 6
UVKZSORBKUEBAZ 6.2 Ki 13 Yes
YLUGVAMRGOIDDQ 6.2 Ki 6
LOCQRDBFWSXQQI 6.2 Ki 16
KLBQZWRITKRQQV 6.2 Ki 21
LNEPOXFFQSENCJ 6.2 Ki 33 Yes
SCZDZQFTMOOIDO 6.2 Ki 6
UNBRKDKAWYKMIV 6.2 Ki 12
DAXNMTILNNCJOI 6.2 Ki 3
GZUITABIAKMVPG 6.2 Ki 22 Yes
HIHZDNKKIUQQSC 6.2 Ki 7
BTYBILKFYYEYRM 6.2 Ki 6
JAXIKFIDJJLTAT 6.2 Ki 6
KLPWJLBORRMFGK 6.2 Ki 8
QSQQQURBVYWZKJ 6.2 Ki 9
WVVSZNPYNCNODU 6.2 Ki 8
BTTOYOKCLDAHHO 6.2 Ki 10
GZKLJWGUPQBVJQ 6.2 Ki 24 Yes
NVDXVBPBFJKQJG 6.2 Ki 3
SVJMLYUFVDMUHP 6.2 Ki 26
SZTNZABXFFPBMM 6.2 Ki 6
YVUQSNJEYSNKRX 6.2 Ki 36
DCSUBABJRXZOMT 6.2 Ki 24
DKGZKTPJOSAWFA 6.2 Ki 21
GPLGAQQQNWMVMM 6.2 Ki 3
UGKUXKJKFRZEQP 6.2 Ki 2
ZEWQUBUPAILYHI 6.2 Ki 21
AHCOOGMIZVMEKD 6.2 Ki 6
DATRLTNBZWRBPI 6.2 Ki 12
MCGZAWFEHFMBAL 6.2 Ki 3
MEZLKOACVSPNER 6.2 Ki 5
OXDMFICMRHFYME 6.2 Ki 6
PNCPYILNMDWPEY 6.2 Ki 13
QSLMDECMDJKHMQ 6.2 Ki 20
XWXCMQFSARGQNK 6.2 IC50 2
UAIBRYGHVVYQBK 6.2 Ki 3
HCWQGDLBIKOJPM 6.1 Ki 12
2D structure