Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
QAESTHCUZJPQGF 6.4 Ki 9
VNSOQQZNVNIEMP 6.4 Kd 3
WJDLKMWEXVEBMK 6.4 Ki 9
YMSCVVXGMWMEMM 6.4 Ki 6
FLMJQBHJNDEDJH 6.4 Ki 6
FXHLGRYCQSRFHY 6.4 Ki 9
HZBAKQLOTJCSJX 6.4 Ki 7
UFFHNEZNXKJHFB 6.4 Ki 10
XIIKDAODIFECTH 6.4 Ki 6
BVWLLEDYRCHASI 6.4 Ki 3
QOYVGASNAZWSTB 6.4 Ki 3
VJUWCGANMBDVKL 6.4 Ki 4
VPFQDYYIEBRWAW 6.4 Ki 3
FEIXCWKYAOFDPF 6.4 Ki 3
HNJJXZKZRAWDPF 6.4 Ki 7
JRNUKVFYILMMLX 6.4 Ki 16
LCKBEOTXTNWYRG 6.4 IC50 8 Yes
FUCGAUZSWYLMRK 6.3 Ki 2
GPVHKTUBAXLWKX 6.3 Ki 3
POCXNIFHHUXWMU 6.3 Ki 3
YQTAOHSPORUWMC 6.3 Ki 5
BOOQTIHIKDDPRW 6.3 Ki 14
CTETYYAZBPJBHE 6.3 Ki 11
DDNAXKKEJCCHMD 6.3 Ki 6
IWHCCXKZMXALTR 6.3 Ki 2
SINCAXCRAGCJEY 6.3 Ki 4
BAZQBEOFVYAFHT 6.3 IC50 5 Yes
BTDBEHJEPKRBOL 6.3 Kd 3
CKLWXPRLRVVKLX 6.3 Ki 3
JTLCTTWVUAIQHD 6.3 IC50 17 Yes
VGKDLMBJGBXTGI 6.3 Ki 7
QWGDMFLQWFTERH 6.3 Ki 23 Yes
VDRGNAMREYBIHA 6.3 Ki 11
YCFVUTASHGKCKL 6.3 Ki 2
MJJALKDDGIKVBE 6.3 IC50 30 Yes
MSQRTETUBFIHMP 6.3 IC50 9 Yes
MWOOWQMUFWOYRV 6.3 Ki 4
ODQWQRRAPPTVAG 6.3 Ki 20 Yes
PAVKAJAAOAJKKE 6.3 Ki 4
RGCVKNLCSQQDEP 6.3 Ki 16
XDRYMKDFEDOLFX 6.3 Ki 13
ANTKBACNWQHQJE 6.3 Ki 12 Yes
BTHSSTHWHHWWSB 6.3 Ki 3
FFRCQBGVCKTCAM 6.3 IC50 2
GDLIGKIOYRNHDA 6.3 Ki 24 Yes
LROGAFKJTOPROQ 6.3 Ki 3
OCBZSBUOYIQXSP 6.3 Ki 6
MDMPKBVNLDREMU 6.3 Ki 3
AFZSMODLJJCVPP 6.3 IC50 12
QVTLLPCYIGXVLX 6.3 Ki 3
2D structure