Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
QRRRICPYXPJYEH 6.6 Ki 2
CWDWGKJQNBEROO 6.5 Ki 3
FZLNIHYBYXMHEO 6.5 Ki 3
IQDINXFLUAYBCC 6.5 Ki 3
JDVBCCBWSXJBJH 6.5 Ki 3
PLDUPXSUYLZYBN 6.5 Ki 22
RDAVKEYAUFGPDX 6.5 Ki 3
RHPCETHLGGFAQB 6.5 Ki 9
WXPNDRBBWZMPQG 6.5 Ki 28
XXJMPUMRHCNWPW 6.5 Ki 8
ACFBDYFNLOKRTR 6.5 Ki 2
OOUPDYBXVFKJRL 6.5 IC50 2
QPXWXQBSYHMBFC 6.5 Kd 3
YMHOBZXQZVXHBM 6.5 Ki 13
ZZJYIKPMDIWRSN 6.5 Ki 11
JFZSEYPHJYDMAZ 6.5 Ki 4
JKDBLHWERQWYKF 6.5 Kd 3
UXABARREKCJULM 6.5 Ki 3
GPZGUIZYGOLWTO 6.5 Ki 6
RNPCOHCWKNMBRI 6.5 Ki 3
YGAFMXXNJBOVBA 6.5 Ki 3
GIJXKZJWITVLHI 6.5 IC50 16
PHLBKPHSAVXXEF 6.5 Ki 12
FYBWLLAUJOWVGO 6.5 Ki 2
XVIIJWXMJCEFCS 6.5 Ki 3
DYPCVKAGDWTSLJ 6.5 Ki 3
HSJYTPFWWPUYDT 6.5 Ki 4
JEZMYAZTGNMODX 6.5 Ki 6
KZVXSSLUUGFVFR 6.5 Ki 14
SMANXXCATUTDDT 6.5 IC50 25 Yes
HTIQEAQVCYTUBX 6.4 IC50 3
KQVZRQLMSQZRDL 6.4 Ki 3
ODLVSMAEEPBMLK 6.4 IC50 2
SIPQEKQXLUBVAY 6.4 Ki 4
BTSCZNWXJQSJIE 6.4 IC50 10
BTSCZNWXJQSJIE 6.4 IC50 10 Yes
FPCCSQOGAWCVBH 6.4 Ki 16
JUQLTPCYUFPYKE 6.4 Ki 25
KMWUPPLGFWGMEM 6.4 Ki 4
RJEWWPFKTYWTSS 6.4 Ki 6
SQEOIKNCNRHYGE 6.4 Ki 6
WEGLOYDTDILXDA 6.4 Ki 22
NTZDCPIPBYWRFF 6.4 IC50 2
RXMGCWHETLRBAF 6.4 Ki 3
SONNWYBIRXJNDC 6.4 Ki 3
CENDKGWAICPCEX 6.4 Ki 2
DLSVKFMVCHCZLY 6.4 Ki 3
HCBLAAMIRQXAHR 6.4 Ki 6
HXHKXXRIQOWOHI 6.4 Ki 3
PQOIDBZLMJMYCD 6.4 Ki 8
2D structure