Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
JJZSKQSMTGTKID 6.7 IC50 2
VUBWIAJSRQTELD 6.7 Kd 3
YHSRTUXPXLVIAG 6.7 IC50 3 Yes
JCCIEQKRVYXDHE 6.7 Ki 4
JXCCNCOVOMQXNP 6.7 Ki 3
HAEPGZUGYMHCJE 6.7 Kd 3
NFQWOMAFZMZYOX 6.7 IC50 5 Yes
HGRHWEAUHXYNNP 6.7 Ki 16
KUWSYGHOSHDWCB 6.7 Ki 3
MGJOAQODMQCCGV 6.7 Ki 3
OZQHHXAYNRRVBN 6.7 Ki 7
TYBWDPQQOPIKEB 6.7 Ki 3
ZKIAIYBUSXZPLP 6.7 Ki 29
FFCFXJXBXUOFIU 6.7 Ki 4
NMTCRDZBJDXVCH 6.7 Ki 5
RRTCFJGKAMKAIY 6.7 Ki 14
IPSCUIDJZTXJJO 6.7 Ki 3
VXOQWXOKZCWYOS 6.7 Ki 2
DVSMVUMYJDOPJQ 6.6 Ki 16
FKKPXTRMLVLGJG 6.6 Ki 7 Yes
GWQQAPMSNKFDFF 6.6 Ki 3
KVWDHTXUZHCGIO 6.6 Ki 32 Yes
VRBKIVRKKCLPHA 6.6 Ki 22
YTBMWHRBVZXATF 6.6 Ki 3
YTJOHEUHUVBKSB 6.6 Ki 3
AVVCHEPXGGYIRM 6.6 Ki 2
GYQWYEJFOYQDMB 6.6 Ki 3
JNBBJUHCODFLEG 6.6 IC50 4
JNMSRIDVZNTYJE 6.6 Ki 2
PHWBOXQYWZNQIN 6.6 IC50 6
LOGUSYSMQQMCJG 6.6 Ki 3
MHNSOBBJZCWUGS 6.6 Ki 17
TTWGDSSADVBNQY 6.6 Ki 12
XXOSLSPHUHLICG 6.6 Ki 3
HUSDORLWRICYQD 6.6 Kd 3
BAADWHDQAKDYLX 6.6 Ki 2
IENZQIKPVFGBNW 6.6 Ki 11 Yes
LGHLMADLDHUIJY 6.6 Ki 7
MVWVFYHBGMAFLY 6.6 Ki 31 Yes
PGGCRGAETLNAJC 6.6 Ki 11
VHFVKMTVMIZMIK 6.6 Ki 15
ZPEIMTDSQAKGNT 6.6 Ki 35 Yes
GSWYYWRNPPQUIJ 6.6 Ki 3
MUHGLPZCYRPXTR 6.6 Ki 3
PGOKBMWPBDRDGN 6.6 IC50 8
LGHLMADLDHUIJY 6.6 Ki 7
LNPDUWGHPCQXJU 6.6 Ki 3
DERZBLKQOCDDDZ 6.6 IC50 20 Yes
DLNKOYKMWOXYQA 6.6 Ki 5
KADUIVAIJUZKJS 6.6 Ki 6
2D structure