Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
DKMFBWQBDIGMHM 6.8 Ki 7
JWIXQLYEPDLLJM 6.8 Ki 7
LNOMHNHLGYHPNB 6.8 IC50 2
OURPZJJZFFKVJH 6.8 Ki 10
RYBOXBBYCVOYNO 6.8 Ki 10
VGUQUIYJFQJLRU 6.8 Ki 9
XJGVXQDUIWGIRW 6.8 Ki 17
ZICGUURZNAJJKQ 6.8 IC50 2
BSOLCASXROXPRZ 6.8 Ki 9
JLVBPZLGXWLQKB 6.8 Ki 8
MTUCTLHCUUYWDV 6.8 Ki 3
AJZBPCAHQHCXMX 6.8 Ki 5
HAEPGZUGYMHCJE 6.8 Kd 3
CDQCFGYTKJPHKT 6.8 Ki 3
CWWOITPDZXNTSJ 6.8 Ki 3
FAIMGWSOSCFGRU 6.8 IC50 6 Yes
IAIZHDGEGFGNMO 6.8 Ki 3
QJUBRJKAGWBYDR 6.8 Ki 5
RNMADLUWJVACLJ 6.8 Ki 9
ADLYXAHODXNVQT 6.8 Ki 5
AUHFSEIMAYONHH 6.8 IC50 2
OGJGQVFWEPNYSB 6.8 Ki 11
PUTAQVRRQAPAQX 6.8 IC50 2
ROUIPNDCVDWYEH 6.8 Ki 2
YNNUSGIPVFPVBX 6.8 Ki 24 Yes
HEDOODBJFVUQMS 6.8 Ki 12
JJCFRYNCJDLXIK 6.8 IC50 25 Yes
SQZSBSSOJVUBRM 6.8 Ki 3
AEDGYKKUCHJGJO 6.8 Ki 3
UREJDUPKGMFJRU 6.8 Ki 17
VGKDLMBJGBXTGI 6.8 IC50 15
XBWUQSHGQYCHAA 6.8 Ki 3
BFKLSSIIDDEGQB 6.7 Ki 2
CQXADFVORZEARL 6.7 Ki 4
HDOZVRUNCMBHFH 6.7 Ki 26 Yes
UKOCGOXTVCIACM 6.7 Ki 13
VSEIJSADDBOANG 6.7 Ki 3
XUSZOVSAUPFWTP 6.7 Ki 3
YJDXDLLDGRBMIT 6.7 Ki 3
ASXGJMSKWNBENU 6.7 Ki 12 Yes
IVEMQVDPOPYVKY 6.7 Ki 2
OGOLMGZJNRNULQ 6.7 Ki 2
VUTLJDGDPMZCOA 6.7 Ki 3
BTDBEHJEPKRBOL 6.7 Kd 3
IYIKLHRQXLHMJQ 6.7 IC50 18
OSEADGVOKYGIER 6.7 Ki 3
HTDIOUCPOHFDQH 6.7 Ki 14
TZFKQPVOFBQHAZ 6.7 Ki 9
GBSLCSDIFSTSOZ 6.7 Ki 4
HEPZPDOHSGVKLD 6.7 Ki 8
2D structure