Target Details
UniProt ACP08913
Gene SymbolADRA2A
Protein NameAlpha-2A adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 761
  • Clinical molecules 54
  • Avg pChEMBL 7.3
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (761)
InChIKey pChEMBL Type Targets Clinical
VWIAFKHHBIYXKV 10.8 IC50 3
MWIKFEVHBBAXIQ 10.8 IC50 3
SWDBYQPERYMOIS 10.5 IC50 3
ZSWAWPHPIFZGTL 10.4 Ki 2
BKRGVLQUQGGVSM 10.3 Ki 18
RCUIZXHMVBJQPJ 10.3 Ki 2
FIERHAFMRVRMDV 10.1 Ki 4
NCOXQFRYWWZGEM 10.0 Ki 3
VGYOOEDZRKNLKS 10.0 Ki 3
YRDASYXEOGTMQU 9.9 IC50 3
ARHWJJBPLJIHQP 9.9 Ki 4
WYFCRYMMLDTJAM 9.8 Ki 4
JKDBLHWERQWYKF 9.7 Kd 3
JKDBLHWERQWYKF 9.7 Kd 3
UCFVOQSSWZQWNE 9.7 Ki 3
GZFYZEHGCPEJAC 9.7 IC50 4
VDSXZDLUEYFJGH 9.7 Ki 4
RTXNZOCMRSFEID 9.6 IC50 4
XQDRWCFJBHLWPR 9.6 Ki 8 Yes
BJNQZYVNKAVYSF 9.6 Ki 6
GKDBTHSYQZTDAJ 9.6 IC50 13
WCIDBLYFACGZGW 9.6 IC50 3
PUJAGVRPJZNJPF 9.5 IC50 4
HPNSJGWCFMHOJX 9.5 IC50 4
JBOWHEDUACRXHK 9.5 Ki 3
JOAHPSVPXZTVEP 9.5 Ki 19
NDIXVNRNAFQAJZ 9.5 Ki 3
XGXYGEYUGTVZAR 9.5 Ki 6
GICQFAWDMCTLDM 9.5 IC50 4
FPQNWBCHCMEAKI 9.5 IC50 4
BRKWIMBSEICBCU 9.4 IC50 4
AYMCTBRVXPCORT 9.4 Ki 3
PRXCUMHAHRIDJF 9.4 Ki 4
DLWKVBPPVYZEML 9.3 Ki 4
FGTWZUQEDNXLLZ 9.3 IC50 4
SYULCMQGHBLEEJ 9.3 Ki 3
UHVQVIBBKZFOBO 9.3 Ki 2
VFIDUCMKNJIJTO 9.3 IC50 4
WDCPMDKQCCZVEW 9.3 Ki 3
AKBJKOBHDJQWMB 9.3 Ki 4
ZYXHQIPQIKTEDI 9.3 IC50 4
ZFZUYTCCHMWWTD 9.2 Ki 9
AKZOIEBLVQLVTR 9.2 IC50 3
JRDUBBHIPPPSLP 9.2 Ki 3
GWAMGWDJCYIREE 9.2 Kd 20
IWBMAAUPHUCYCI 9.2 Kd 20
MODBIBJHAWXYOZ 9.2 Kd 20
WLWNODXEXGTHDO 9.2 IC50 4
ZRQMUCDHVVOENY 9.2 Kd 17
WVDIRTLHBANRPM 9.2 IC50 3
2D structure