Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
GLRXSDVYMJTKAU 6.4 Ki 4
JNBDSWBJCGQGPV 6.4 Ki 5
UUQSWYMJKUSTBX 6.4 Ki 5
ATALOGFLLWJSLP 6.4 Ki 2
DATRLTNBZWRBPI 6.4 Ki 12
FPGYVSKEOKZERL 6.4 Ki 5
HSHUYRPIECSXLE 6.4 IC50 4
MPVIJPUSNDEBBO 6.4 Ki 5
HRIDJFHKBNVJDP 6.4 Ki 5
KYIAOTGZEXVAKQ 6.4 Ki 2
MOXAZUHAPUILEZ 6.4 Ki 3
UNZBDOQVZFAUNP 6.4 Ki 5
IVUOMTRDHAJWCR 6.4 IC50 4
OJSFTALXCYKKFQ 6.4 Ki 10
BFKVAWMWDMHLEZ 6.4 Ki 5
FIMOHMGQXMTFNO 6.4 IC50 5
IENFGCJKCCNIMB 6.4 Ki 5
TWMKVARMUAJVEO 6.4 Ki 2
BYOZMAAKKNZOCN 6.4 Ki 5
CHSDYWULPTYCTA 6.4 Kd 5
FPTVPLUMEFOZHQ 6.4 Ki 4
ZUSQEIFGHOIMSY 6.4 Ki 5
LGCNGBKZRRQUBB 6.4 Ki 5
VGKDLMBJGBXTGI 6.4 IC50 15
VGSYEFOBFMUWGO 6.4 Ki 6
VLPCMABIYZTMKT 6.4 Ki 2
YSPKJODQLIOHOF 6.4 Kd 5
HCVAFIOQGLGPAZ 6.3 Ki 5
SAPNXPWPAUFAJU 6.3 Ki 10
UFOTTYHVWBYOKX 6.3 Ki 5
GEULRCAVYVOGLC 6.3 Ki 2
KSNHHKZYKYNBEI 6.3 Ki 6
MVNBPMNELMRFMU 6.3 Ki 5
NWMFUMWLMFJZLH 6.3 IC50 5
UUQSWYMJKUSTBX 6.3 Ki 5
ATMXUFMBNANYLL 6.3 Ki 5
GCMYOOAJYOMGJH 6.3 Ki 5
LRBPZOOGQFAYKA 6.3 Kd 5
RWZFXPOJQFVTQX 6.3 IC50 3
FMPNFDSPHNUFOS 6.3 Ki 5
FMPNFDSPHNUFOS 6.3 Ki 5
UREJDUPKGMFJRU 6.3 Ki 17
ARRNZUHFFUCBML 6.3 IC50 4
CTPZAQGPYTYXAV 6.3 Kd 5
FPDIERBPQFAFSI 6.3 Ki 17 Yes
RAVGDLZWTLVAPH 6.3 Ki 5
XCSJIKDLUXGHQG 6.3 Ki 4
ZMDYOFHOFRJYRX 6.3 IC50 3
HPXSCBIGYJMQQH 6.3 Ki 5
RGKNMWKLNOOSDH 6.3 IC50 5
2D structure