Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
HDOZVRUNCMBHFH 6.6 Ki 26 Yes
RNNZREWYEVVFIS 6.6 IC50 4
RQDLDNLBJUDOFV 6.6 Ki 4
BDKHSETYUSIWLB 6.6 Ki 3
GUYHTHYSWVZNOT 6.6 Ki 3
PKQJAHUVAHVQSO 6.6 Ki 5
WQEUCWAEHCWTPL 6.6 Ki 3
YPUMMBFUPIPODG 6.6 IC50 5
UEQUQVLFIPOEMF 6.6 IC50 21 Yes
ZCVMWBYGMWKGHF 6.6 Ki 19 Yes
RTVAKAAPGHVGBW 6.6 Ki 5
ZQIYKYBVHCNJMX 6.6 IC50 5
JRNKPQVEBTTXNH 6.5 Kd 5
MWDWETWIXZBNRI 6.5 Ki 2
SXWJLTLRDSROPE 6.5 Ki 2
MJJALKDDGIKVBE 6.5 IC50 30 Yes
NASFNLMUWVJIEY 6.5 Ki 5
UNZBDOQVZFAUNP 6.5 Ki 5
VGSSLDYPUXVRJF 6.5 Ki 2
XFBTXTHJTCSANR 6.5 Ki 5
HTKBZSOYVFEBSC 6.5 Ki 5
PCWGGOVOEWHPMG 6.5 Ki 12
ROCCLUYSPSAIDK 6.5 Ki 5
BSSWNYCCQZRJSB 6.5 Ki 5
CZWQBSKNHUVZLI 6.5 IC50 5
VPWKHNIBDCHPNN 6.5 Ki 5
BFELQLHLUNQIHL 6.5 Ki 5
BTTOYOKCLDAHHO 6.5 Ki 10
DTDHZMMUUQJYIO 6.5 Ki 5
QOMMMTAFQPGRCW 6.5 Ki 5
KQHKTHFVDIBYJZ 6.5 Ki 5
LOAZWNRCWBWKAC 6.5 Ki 5
RPMBYDYUVKEZJA 6.5 Ki 8
UOGBSPSWAMZQNS 6.5 IC50 2
UZJWAFOJOSGEKL 6.5 IC50 15
FHPIXVHJEIZKJW 6.5 Ki 18 Yes
LOZFSJRXJHXNTK 6.5 IC50 3
NYNKCIGJEUJVIL 6.5 IC50 2
OXWXUIXTFQJYIL 6.5 Ki 5
CRXJTADTDFNFTC 6.5 IC50 5
GPZMWOXSIRVXQW 6.5 Ki 8
ZOEYTLRCDGNMCU 6.5 Ki 5
ABRYVCKEQWCHSC 6.5 Ki 5
ATQMRMGXINTJHV 6.5 Ki 9 Yes
GKFAOGATDDYRDQ 6.5 Ki 5
WKEGMVFSZKEMJV 6.5 Ki 5
FRSBYJSARNVZCX 6.5 Ki 5
QCSKQMQBRQOXLU 6.5 Ki 5
QHFVUCATFKHMCG 6.5 Ki 5
BRBVBRCNTVSDRI 6.4 Ki 2
2D structure