Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
VBTYLZVMQCAWDY 6.8 Ki 4
WULCBOSTMCYKCZ 6.8 Kd 5
AZYYVQIBCPFAIG 6.8 Ki 5
YUCQRSFKFKVEJX 6.8 IC50 4
JCBGAEQLPPOPDK 6.8 Ki 5
XFRRXQDVSCYLBU 6.8 Ki 5
XJFLDBYRKJAMIK 6.8 Ki 5
UWKMFEOQWPCWLU 6.7 Ki 5
WIKYUJGCLQQFNW 6.7 IC50 23 Yes
CPJMEEZDGWZNFW 6.7 Ki 2
IEUILNNAXQDVCX 6.7 Ki 3
JRXSQQHZULYLDJ 6.7 IC50 3
LBMILISNRUJASD 6.7 Ki 2
PBCNZXLLSIAHHR 6.7 Ki 2
GRHQYMDSSBRZTL 6.7 Kd 5
MNTJDNKIZZJMSD 6.7 IC50 5
KUKJOLRCPDCJAJ 6.7 Ki 5
MRTRSVIAPJHYNC 6.7 Kd 5
OUQAVICYOCWJLG 6.7 Ki 5
VHYUYQHTMPWAPK 6.7 Kd 5
MVDUBVLGXGZDSV 6.7 Ki 4
STUWFURQGSMWES 6.7 Ki 5
CUCVCEWRTFMXDA 6.7 IC50 5
LRBPZOOGQFAYKA 6.7 Kd 5
GMLQVLRORNVELR 6.7 Ki 5
GZRIGDJQQNOXAM 6.7 IC50 5
KSKFIMPGQOTLKR 6.7 Ki 5
VPWKHNIBDCHPNN 6.7 Ki 5
AVNRDCQRRUOTCC 6.6 Ki 5
HLFXMJFGYOOILI 6.6 Ki 3
VUCYYOGBXRCVIJ 6.6 Ki 5
WKEGMVFSZKEMJV 6.6 Ki 5
ZSEXCDQYDWJYHN 6.6 Ki 5
ZZVUWRFHKOJYTH 6.6 Ki 11 Yes
DPSJSZQSAMCEEQ 6.6 IC50 5
QOJBMAYEUGMTTA 6.6 Ki 5
DLMOQVWYEFDOHH 6.6 Ki 5
MYODZQJNSSBKEB 6.6 Ki 3
VHYUYQHTMPWAPK 6.6 Kd 5
WMGWWIZDKKAUOR 6.6 Ki 3
WTWPGUIYLXNGRX 6.6 Ki 5
XJGVXQDUIWGIRW 6.6 Ki 17
FTFRVHRVNAJZCB 6.6 Ki 5
HNLUMKGZTQUVEY 6.6 Ki 5
JAUOIFJMECXRGI 6.6 IC50 13
IMKYINSUEJXTJZ 6.6 Ki 5
NWZNQDANKXXDFA 6.6 Ki 5
PUNXWODWMDLZDP 6.6 Ki 5
YIDUXCASAXKJEC 6.6 Ki 5
FVMATSHOWXOARI 6.6 IC50 2
2D structure