Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
DGWWXFCHEOPTQT 7.0 Ki 3
IBZJKEOJOGAMGJ 7.0 Ki 11 Yes
PGDYOGMNQCUWMZ 7.0 Ki 5
XYIJOTOXQIJOIN 7.0 Kd 5
QTQLWKLZSPZQTO 7.0 Ki 5
FHJHJYBFXRHWSS 7.0 Ki 4
GTXZQPRWWKNJQL 7.0 Ki 5
HECAWZFPXYNICY 7.0 Ki 5
KKEGQSSUXOGEAF 7.0 Ki 5
KBFDMWOMIBRCFI 7.0 Ki 2
QRUXDRCXIGZTGT 7.0 Ki 5
VUWOKTOQKPRPDM 7.0 Ki 5
WULCBOSTMCYKCZ 7.0 Kd 5
HTYJHPPHBQRXGX 7.0 Ki 5
LISJYMSYSGWFLD 7.0 Ki 5
HBLWDHBKUANPEG 6.9 IC50 5
RHAFROHARIZTPJ 6.9 Kd 5
SIYLLGKDQZGJHK 6.9 IC50 13
FPUKGJMTLUQGFZ 6.9 Ki 12
NSIYNGOBBBLDIU 6.9 Ki 2
VBPQNYMWBQALHS 6.9 Ki 5
WCQIGWGZUOSGET 6.9 Ki 5
WXXOCGISBCTWPW 6.9 Ki 4
AHOUBRCZNHFOSL 6.9 Ki 13
XKYMIJTXUGXDLR 6.9 Ki 4
RMHMFHUVIITRHF 6.9 Ki 5
XCYNAFSXKQRKGO 6.9 Ki 5
JGOLLLMMDGFRBE 6.9 Ki 4
QCKCTTSCZBLBGX 6.9 Ki 3
AILVCKQCTVDJPU 6.9 Ki 4
BNMMMFMJYKFYRQ 6.9 Kd 5
IEEFWRMSEALUNN 6.9 Ki 5
QSLMDECMDJKHMQ 6.9 IC50 20
CPHUSFMAHLLFQS 6.9 IC50 5
CLKYBOTWHCENMP 6.8 Ki 5
PIBNOUQILXRVNG 6.8 Ki 5
WYXGHKGJTWRLPO 6.8 Ki 2
HCYAFALTSJYZDH 6.8 Ki 14 Yes
KHLGLAZJVORACT 6.8 Ki 3
PGZUAZYZPAOAOH 6.8 Ki 2
QZTQQKQHRWQZMZ 6.8 Ki 4
UCBXWLPRAVDTBU 6.8 Ki 5
XINSCWBHVQVKQT 6.8 Kd 5
YAUZNKLMKRQDAM 6.8 Ki 7
HXQMZFUQSGJNPQ 6.8 Ki 5
JETRJUTXVVSGTR 6.8 Ki 4
SADFFAQSWHTWLL 6.8 Ki 5
WDLCZGMJXFWVAF 6.8 IC50 4
XCYWQSIELKTIEB 6.8 Ki 5
UWQNUCNXNKMWKG 6.8 Ki 5
2D structure