Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
FJOQSAAWJBXPCK 7.2 Ki 5
SLVMESMUVMCQIY 7.2 Ki 14
WEVVZJGQIWKFOJ 7.2 Ki 2
WMPSFVBNWOMJKI 7.2 Ki 3
DZSCHRPHQBQAFZ 7.2 IC50 5
NHUURXLCGOCXHZ 7.2 Ki 5
QPNVVIACYJVUOX 7.2 Ki 12
QTBCATBNRIYMPB 7.2 Ki 5
SKEKXGMFLBCYNC 7.2 Ki 5
XMDRTFUFPOAGDR 7.2 Ki 9
GNHXYBDOJNQUSM 7.2 Ki 4
UFUQREONAQKXQA 7.2 Ki 5
YZCWHHFUBMQIKE 7.2 Ki 5
JDCADUVEQJRIDC 7.2 Ki 5
UOKGNINOAYOIDX 7.2 Ki 5
LYFQHKXGGDVXCQ 7.2 Ki 5
NXIFJNOHOQFSCE 7.1 Ki 5
WIEMOFKMOGPXQF 7.1 Ki 5
ZPMRLGPLMNVIDC 7.1 Ki 4
BGDKAVGWHJFAGW 7.1 IC50 7
GQAHLUHWIIZPFR 7.1 Ki 5
IJRUGZIZSARHLR 7.1 Ki 5
ODQWQRRAPPTVAG 7.1 Ki 14
AESSYHBGSGYEPG 7.1 Ki 5
GZEKHKZVPHPQCL 7.1 Ki 5
ICZVKTVMHVHOQI 7.1 Ki 5
PBHNZQQGQQOYNM 7.1 IC50 5
DSPDJPFEBQTXDO 7.1 Kd 5
NBNHGRRWKSPRMB 7.1 Ki 2
TZADATSLTAFDKI 7.1 Ki 3
DKVRRZMTJBDMTP 7.1 IC50 3
OANBYDFPBWKVGI 7.1 Ki 5
BCGWQEUPMDMJNV 7.1 Ki 30 Yes
ILHSFCNKNNNPRN 7.1 Ki 3
FNNCHHONWUGPND 7.1 IC50 5
VMJKUCKTXMESQR 7.1 Ki 5
DMQAXIJUTYJHIV 7.1 Ki 6
PSOFWCMIGQGVAZ 7.1 Ki 2
LVKGEHAPRFNGNI 7.0 Kd 5
OHEDKBMQRCAABJ 7.0 IC50 6
PHTUQLWOUWZIMZ 7.0 Ki 7
BZCOASIWPFVBQZ 7.0 Kd 5
RVTKNIPUELNCNR 7.0 Ki 5
AKPOTJIMZXGFLY 7.0 Ki 5
PTBANFXYQIIDAF 7.0 Ki 5
CHXGLJOIUDBPTI 7.0 Ki 5
DSPDJPFEBQTXDO 7.0 Kd 5
NZUPCNDJBJXXRF 7.0 Ki 5
XLHVWZIVNKAJOS 7.0 IC50 5
AKPSMQSQINOOPH 7.0 Ki 5
2D structure