Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
UBGMVJXVELKNMU 7.5 Ki 5
UPDOKFNDDXFBCH 7.5 Ki 4
VYVYCDJDMPVQTH 7.5 Ki 2
CUYJUFFZSFIMQM 7.5 Ki 5
FNCJWKNHUAURLL 7.5 Ki 5
KFMIEAZKENMLEL 7.5 Ki 5
QFRDMVXRTJXQSC 7.5 Ki 5
QGJWMGIPVUWDAK 7.5 Ki 5
OFBOKKRZVJJZHR 7.5 Ki 5
ZPEIMTDSQAKGNT 7.5 Ki 35 Yes
CJRUIOCIHPGNQL 7.5 Ki 5
XFGSFWFIJFNGQY 7.5 Ki 5
YUJOQEAGGUIMED 7.5 Ki 5
DIDYGLSKVUKRRP 7.5 Ki 5
SLFGIOIONGJGRT 7.5 Ki 12
XPXPKUQRUOKHFD 7.5 Ki 5
RHAFROHARIZTPJ 7.5 Kd 5
LPJZXUYTCJIHTG 7.4 Ki 5
VWBQUAMKHIBZSG 7.4 Ki 5
KOKXORZIPKJNJL 7.4 Ki 5
DJIVSTFQGOLPFP 7.4 Ki 4
GZIIELZICVUEPK 7.4 Ki 5
JOLJIIDDOBNFHW 7.4 Ki 14
UKIPQWNRWJEJMN 7.4 Ki 4
VPWKHNIBDCHPNN 7.4 Ki 5
QJBDLOQOXGQJTD 7.4 Ki 5
USWIIRIGMDFSNJ 7.4 IC50 5
FBOUYBDGKBSUES 7.4 Ki 6
GDLIGKIOYRNHDA 7.3 IC50 24 Yes
PMCCMEISWXQOME 7.3 Kd 5
HTYJHPPHBQRXGX 7.3 Ki 5
ZTVIKZXZYLEVOL 7.3 IC50 5
HNJAEIXPTNJDDI 7.3 Ki 5
XPXPKUQRUOKHFD 7.3 Ki 5
LOOAMMHLLVGAEL 7.3 Ki 5
JNNOSTQEZICQQP 7.3 Ki 7
KWBBYHOSQKDRRU 7.3 Ki 3
LACUGMNHRWEZND 7.3 Ki 5
NFVADXLLOOOZIS 7.3 Ki 5
OMOWOTRKFFNAIT 7.3 IC50 5
UFSZYKLBZJNXLV 7.3 Ki 5
WHZBQLWHOPDIPC 7.3 Ki 5
YRIHWSWKYBUXOL 7.2 IC50 5
TWCQJLAORZMNFA 7.2 IC50 5
ZNXQAFLLESPBNZ 7.2 Ki 5
AYQKIBOBFAZBCX 7.2 Ki 5
MCMLNRXJLVBKFA 7.2 Ki 4
UNZBDOQVZFAUNP 7.2 Ki 5
YKICXCKVEJORPH 7.2 Ki 5
BLFDLFBLCZXAQW 7.2 Ki 4
2D structure