Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
OYXCACHCXKHEOC 8.0 Ki 5
KHJKTXKHUACAIJ 8.0 Ki 5
PHRZGNXUUFTVSE 8.0 Ki 5
PHRZGNXUUFTVSE 8.0 Ki 5
HWHLPVGTWGOCJO 8.0 Ki 6
ZMDWHSSHCTZQTD 8.0 Ki 5
BZHQFTZHZVTIMQ 8.0 Ki 5
GZXQKCMKEJCSMK 8.0 Kd 5
JYKJJNTVFIWSHT 8.0 Kd 5
ONOZLVJQXQZLPL 8.0 Ki 5
UXRUOZRDTXTVAI 8.0 Ki 5
ZUXABONWMNSFBN 8.0 Ki 29
AVNRDCQRRUOTCC 7.9 Ki 5
AYFAGRAOJPSHSH 7.9 Ki 19
AVNRDCQRRUOTCC 7.9 Ki 5
PXHIFOLPKHLYBX 7.9 Ki 5
KLBQZWRITKRQQV 7.9 Ki 21
ITDUNAGUAFBFRA 7.8 Ki 5
SNSMIIQEKVYNOH 7.8 Ki 5
YNNUSGIPVFPVBX 7.8 Ki 24 Yes
OGTLDFSTCJABJV 7.8 Ki 5
MEAOYGFCVURJIU 7.8 Kd 5
FFWZAKHCGSHEHR 7.8 Ki 2
IZPDHAHWQOHFNJ 7.8 Ki 2
OBWGMKKHCLHVIE 7.8 Ki 9
WXPNDRBBWZMPQG 7.8 Ki 28
WHKGYJCRLQITBW 7.8 Ki 5
WHKGYJCRLQITBW 7.8 Ki 5
POIIDLJXIAHDFT 7.8 Ki 5
UWVWASPAVBANND 7.8 Ki 5
HTYJHPPHBQRXGX 7.7 Ki 5
ICDMIDKSZQHGHA 7.7 Ki 2
BRMKEVBAZDNRPY 7.7 Kd 5
IXXCPZGOFVCPCH 7.7 Ki 5
GHJAWSFCIDDAHY 7.7 Ki 2
OTYJWRFICHGQJT 7.7 Ki 5
QZUDBNBUXVUHMW 7.7 Ki 39 Yes
UFSZYKLBZJNXLV 7.7 Ki 5
ODQWQRRAPPTVAG 7.7 IC50 20 Yes
DJOCICQNBMTMNG 7.6 Ki 5
WYDUSKDSKCASEF 7.6 Ki 5
GFDOCHMSKUCLIW 7.6 Ki 5
UNZBDOQVZFAUNP 7.6 Ki 5
VQMYCZUUGWZZTK 7.6 IC50 5
MVNBPMNELMRFMU 7.6 Ki 5
QVYRGXJJSLMXQH 7.5 Ki 14
KVWDHTXUZHCGIO 7.5 Ki 32 Yes
UPPMZCXMQRVMME 7.5 IC50 7
PMNZXPJWRDBQSA 7.5 Ki 5
POGDAPYUQHRUOU 7.5 Ki 5
2D structure